SCHEMBL2774544

SCHEMBL2774544

Cc1ccc(S(=O)(=O)C2CCN(CCc3ccc4occc4c3)C2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.43
KCNH2 Q12809 5/20 0.43
HTR2C P28335 4/20 0.43
CA12 O43570 3/20 0.41
CA2 P00918 3/20 0.41
CA1 P00915 2/20 0.41
CA4 P22748 2/20 0.41
CA5A P35218 2/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41
CA13 Q8N1Q1 2/20 0.41
CA14 Q9ULX7 2/20 0.41
NAMPT P43490 2/20 0.38
KCNQ1 P51787 1/20 0.37
CHRM5 P08912 2/20 0.36
DRD2 P14416 2/20 0.36
CTNNB1 P35222 1/20 0.36
WNT3A P56704 1/20 0.36
HTR1A P08908 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2774034 0.86 HTR1A (0.40) HTR2AKCNH2HTR2CCA12CA2
SCHEMBL2776295 0.81 HTR1A (0.38) HTR2AKCNH2HTR2CCA12DRD2
SCHEMBL22634126 0.78 HTR2A (0.70) HTR2AKCNH2HTR2CCA12CA2
SCHEMBL2775792 0.77 CHRM5 (0.52) HTR2AKCNH2HTR2CCA12CA2
SCHEMBL2775632 0.76 HRH3 (0.39) KCNH2CA12CA2CHRM5HTR1A
SCHEMBL2775113 0.75 HTR1A (0.42) KCNH2HTR1ACYP2D6SLC6A4
SCHEMBL2774320 0.75 HRH3 (0.54) KCNH2HTR1ACYP2D6SLC6A4
SCHEMBL2773779 0.72 DRD2 (0.40) KCNH2DRD2HTR1ACYP2D6SLC6A4
SCHEMBL7022479 0.72 HTR2A (0.63) HTR2AKCNH2HTR2CCA12CA2
SCHEMBL14033350 0.69 HRH1 (0.46) HTR2AKCNH2KCNQ1CHRM5DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010112488-A1 METHOD FOR OBTAINING 1,3-DIFUNCTIONALIZED PYRROLIDINE DERIVATIVES RAGACTIVES, S.L.U. (ES) 2010-10-07 WO claimed
EP-2236509-A1 Method for obtaining 1,3-difunctionalized pyrrolidine derivatives Ragactives, S.L. (ES) 2010-10-06 EP claimed
WO-2010112488-A1 METHOD FOR OBTAINING 1,3-DIFUNCTIONALIZED PYRROLIDINE DERIVATIVES RAGACTIVES, S.L.U. (ES) 2010-10-07 WO disclosed
EP-2236509-A1 Method for obtaining 1,3-difunctionalized pyrrolidine derivatives Ragactives, S.L. (ES) 2010-10-06 EP disclosed