SCHEMBL2775632

SCHEMBL2775632

CS(=O)(=O)OC1CCN(CCc2ccc3occc3c2)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.39
CA2 P00918 2/20 0.38
CA12 O43570 1/20 0.38
HTR1A P08908 4/20 0.38
CYP2D6 P10635 3/20 0.38
SLC6A4 P31645 3/20 0.38
ROCK2 O75116 1/20 0.37
ESR1 P03372 1/20 0.35
CHRM4 P08173 1/20 0.35
KCNH2 Q12809 1/20 0.35
MCHR2 Q969V1 1/20 0.35
MCHR1 Q99705 1/20 0.35
HTR1B P28222 2/20 0.34
CHRNA1 P02708 2/20 0.34
CHRNG P07510 2/20 0.34
CHRNB1 P11230 2/20 0.34
CHRNB2 P17787 2/20 0.34
CHRNB4 P30926 2/20 0.34
CHRNA3 P32297 2/20 0.34
CHRNA7 P36544 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2773779 0.87 DRD2 (0.40) HTR1ACYP2D6SLC6A4ROCK2ESR1
SCHEMBL2774034 0.84 HTR1A (0.40) HRH3CA2CA12HTR1ACYP2D6
SCHEMBL2774320 0.79 HRH3 (0.54) HRH3HTR1ACYP2D6SLC6A4ROCK2
SCHEMBL6796403 0.78 ADRA1D (0.47) HRH3HTR1ASLC6A4MCHR1
SCHEMBL2775113 0.77 HTR1A (0.42) HRH3HTR1ACYP2D6SLC6A4ROCK2
SCHEMBL6796681 0.77 L3MBTL1 (0.49) HRH3HTR1ASLC6A4KCNH2
SCHEMBL2776295 0.77 HTR1A (0.38) HRH3CA12HTR1ACYP2D6SLC6A4
SCHEMBL2774544 0.76 HTR2A (0.43) CA2CA12HTR1ACYP2D6SLC6A4
SCHEMBL6802876 0.76 SIGMAR1 (0.55) HRH3HTR1ASLC6A4KCNH2
SCHEMBL2776390 0.76 SLC6A4 (0.54) HRH3HTR1ACYP2D6SLC6A4CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010112488-A1 METHOD FOR OBTAINING 1,3-DIFUNCTIONALIZED PYRROLIDINE DERIVATIVES RAGACTIVES, S.L.U. (ES) 2010-10-07 WO disclosed
EP-2236509-A1 Method for obtaining 1,3-difunctionalized pyrrolidine derivatives Ragactives, S.L. (ES) 2010-10-06 EP disclosed