SCHEMBL27749033

SCHEMBL27749033

CNc1c(Cl)cc(C(F)(F)F)cc1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.41
TACR1 P25103 7/20 0.41
GABRA2 P47869 2/20 0.40
GABRB2 P47870 2/20 0.40
ACLY P53396 3/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MET P08581 2/20 0.39
GABRP O00591 1/20 0.39
GABRD O14764 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27727995 0.83 METAP2 (0.42) METAP2TACR1ACLYMETKIF11
SCHEMBL1768628 0.79 PDE2A (0.40) GABRA2GABRB2MAPTSMN1; SMN2GABRP
SCHEMBL27926226 0.73 GRM2 (0.52) GABRA2GABRB2NPC1MAPTNFKB1
SCHEMBL28806082 0.73 KIF11 (0.52) METAP2NPC1MAPTNFKB1RAB9A
SCHEMBL27749081 0.73 PLK1 (0.38) TACR1ACLY
SCHEMBL28320613 0.72 KIF11 (0.47) METAP2TACR1MAPTKIF11BACE1
SCHEMBL2139259 0.72 KIF11 (0.50) METAP2TACR1GABRA2GABRB2ACLY
SCHEMBL10280738 0.71 GABRA2 (0.38) GABRA2GABRB2MAPTSMN1; SMN2GABRP
SCHEMBL7715418 0.71 ALDH1A1 (0.47) MAPTRAB9ASMN1; SMN2
SCHEMBL27720555 0.69 METAP2 (0.50) METAP2TACR1METKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101331124-B Novel capsaicin receptor ligands and their use for the manufacture of medicaments GRUENENTHAL GMBH 2013-08-14 CN disclosed
CN-101331124-A Novel capsaicin receptor ligands and their use for the manufacture of medicaments GRUENENTHAL CHEMIE (DE) 2008-12-24 CN disclosed