SCHEMBL27749079

SCHEMBL27749079

CNc1cc(F)c(C(F)(F)F)cc1-c1ccccc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 6/20 0.40
GPR3 P46089 1/20 0.40
AR P10275 1/20 0.40
CYP3A4 P08684 3/20 0.37
CYP1A2 P05177 2/20 0.37
DHODH Q02127 1/20 0.37
MAT2A P31153 2/20 0.36
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP2C19 P33261 2/20 0.34
CYP2D6 P10635 1/20 0.34
ALOX15 P16050 1/20 0.34
MAPK1 P28482 1/20 0.34
HSD17B10 Q99714 1/20 0.34
STK10 O94804 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27749032 0.76 HSD11B1 (0.46) HSD11B1GPR3MAT2AALDH1A1KDM4E
SCHEMBL9231954 0.71 MEN1 (0.38) GPR3ARMEN1KMT2AALOX15
Hydrochloric Acid SCHEMBL28453942 0.70 MEN1 (0.37) GPR3ARALDH1A1MEN1KMT2A
SCHEMBL6862522 0.69 CYP2A6 (0.44) HSD11B1CYP3A4CYP1A2DHODHALDH1A1
SCHEMBL1262778 0.69 HSD11B1 (0.59) HSD11B1ARCYP3A4ALDH1A1KDM4E
SCHEMBL20329695 0.69 TDP1 (0.41) HSD11B1CYP3A4CYP1A2ALDH1A1KDM4E
SCHEMBL28828302 0.68 HSD11B1 (0.50) HSD11B1GPR3ARALDH1A1KDM4E
SCHEMBL9233334 0.68 KIF11 (0.38) GPR3ARMEN1KMT2AALOX15
SCHEMBL9232865 0.67 KDR (0.35) ARMEN1KMT2AALOX15MAPK1
SCHEMBL9281931 0.66 APP (0.40) ARCYP3A4CYP1A2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101331124-B Novel capsaicin receptor ligands and their use for the manufacture of medicaments GRUENENTHAL GMBH 2013-08-14 CN disclosed
CN-101331124-A Novel capsaicin receptor ligands and their use for the manufacture of medicaments GRUENENTHAL CHEMIE (DE) 2008-12-24 CN disclosed