SCHEMBL27752111

SCHEMBL27752111

O=CC(CBr)c1ccc(Cl)s1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 1/20 0.39
GABBR1 Q9UBS5 1/20 0.39
GSK3B P49841 1/20 0.32
WRN Q14191 1/20 0.31
F2 P00734 1/20 0.31
DAO P14920 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27893994 0.83 GABBR2 (0.40) GABBR2GABBR1GSK3BWRNF2
SCHEMBL27708206 0.79 GSK3B (0.36) GSK3BWRNDAO
SCHEMBL27586775 0.78 ALOX5 (0.37) DAO
SCHEMBL27708354 0.78 WRN (0.31) WRN
SCHEMBL27804136 0.75 WRN (0.37) WRN
SCHEMBL1849742 0.75 GABBR2 (0.39) GABBR2GABBR1GSK3BWRNF2
SCHEMBL27894259 0.74 LMNA (0.37) GABBR2GABBR1
SCHEMBL7067216 0.72 GABBR2 (0.40) GABBR2GABBR1GSK3BWRNF2
SCHEMBL27616109 0.71
SCHEMBL4706414 0.71 GABBR2 (0.39) GABBR2GABBR1GSK3BWRN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102791714-A N-(imidazopyrimidin-7-yl)-heteroarylamide derivatives and their use as PDE10A inhibitors HOFFMANN LA ROCHE 2012-11-21 CN disclosed
CN-102112474-A Quinuclidine carbonate derivatives and medicinal composition thereof CHIESI FARMA SPA 2011-06-29 CN disclosed
CN-102056907-A Heterocyclic derivative and use thereof TAKEDA PHARMACEUTICAL 2011-05-11 CN disclosed
CN-101511429-A Indulines derivatives and gpr119 agonists SMITHKLINE BEECHAM CORP (US) 2009-08-19 CN disclosed