SCHEMBL2775288

SCHEMBL2775288

COC(=O)c1ccc(-c2cnc(CCC(O)c3ccc(Oc4ccccc4)cc3)o2)nc1

nearest known ligand 0.61

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
FAAH O00519 4/20 0.49
CES1 P23141 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2774812 0.90 FAAH (0.49) FAAHCES1
SCHEMBL2775285 0.83 FAAH (0.59) FAAHCES1
SCHEMBL2776361 0.76 FAAH (0.73) FAAHCES1
SCHEMBL2774807 0.75 FAAH (0.58) FAAHCES1
SCHEMBL29596790 0.73 RXFP1 (0.56)
SCHEMBL2772835 0.69 CES1 (0.67) FAAHCES1
SCHEMBL2776228 0.68 FAAH (0.75) FAAHCES1
SCHEMBL28106567 0.68 LMNA (0.61)
SCHEMBL2774811 0.67 FAAH (0.72) FAAHCES1
SCHEMBL2772700 0.66 FAAH (0.77) FAAHCES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2152082-A1 TETRACYCLIC INHIBITORS OF FATTY ACID AMIDE HYDROLASE The Scripps Research Institute (US) 2010-02-17 EP disclosed
WO-2008147553-A1 TETRACYCLIC INHIBITORS OF FATTY ACID AMIDE HYDROLASE THE SCRIPPS RESEARCH INSTITUTE (US) 2008-12-04 WO disclosed