SCHEMBL27753602

SCHEMBL27753602

Nc1cc(CN(Cc2ccccc2)OC(=O)Cc2ccccc2)ccc1OCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
FOLH1 Q04609 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
FFAR1 O14842 1/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
LTB4R Q15722 2/20 0.39
LTB4R2 Q9NPC1 2/20 0.39
APP P05067 1/20 0.38
PTGER1 P34995 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4643523 0.78 MEN1 (0.45) ALOX5MEN1KMT2AFOLH1FFAR4
SCHEMBL6079992 0.73 APP (0.50) FOLH1L3MBTL1MAPK1FFAR4FFAR1
SCHEMBL11085556 0.73 KDM4E (0.50) MEN1KMT2AL3MBTL1ALDH1A1
SCHEMBL16300892 0.72 APP (0.46) FOLH1L3MBTL1MAPK1FFAR4FFAR1
SCHEMBL10410151 0.71 ALOX5 (0.52) ALOX5FOLH1FFAR4LTB4RLTB4R2
SCHEMBL5783643 0.71 APP (0.47) KMT2AFOLH1L3MBTL1MAPK1FFAR4
SCHEMBL8057639 0.70 LMNA (0.52) MEN1KMT2AFOLH1L3MBTL1ALDH1A1
Acetic Acid SCHEMBL9653704 0.70 SMN1; SMN2 (0.52) FOLH1L3MBTL1ALDH1A1CYP2C19FFAR4
SCHEMBL10409146 0.69 APP (0.49) L3MBTL1FFAR4FFAR1APP
SCHEMBL2009073 0.69 CREBBP (0.66) MEN1KMT2AL3MBTL1ALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101321743-A 1,1, 3-trioxo-1, 2, 5-thiadiazolidines as PTP-enzyme inhibitors and their use NOVARTIS AG (CH) 2008-12-10 CN disclosed