SCHEMBL27760176

SCHEMBL27760176

COc1ccccc1CNc1ncnc2c1ccn2C1C[CH]C(O)C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.53
LMNA P02545 5/20 0.51
TP53 P04637 3/20 0.51
MAPT P10636 2/20 0.51
MAPK1 P28482 5/20 0.49
POLB P06746 1/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
TNF P01375 1/20 0.48
NOD1 Q9Y239 1/20 0.48
ADORA3 P0DMS8 1/20 0.47
ADORA2A P29274 1/20 0.47
ADORA1 P30542 1/20 0.47
ALDH1A1 P00352 7/20 0.47
TSHR P16473 7/20 0.47
HSD17B10 Q99714 6/20 0.47
CYP1A2 P05177 5/20 0.47
CYP3A4 P08684 5/20 0.47
CYP2D6 P10635 5/20 0.47
CYP2C19 P33261 5/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27739696 0.85 AURKA (0.45) ADORA3ADORA2AADORA1AURKARPS6KB1
SCHEMBL5456441 0.84 KDM4E (0.52) KDM4ELMNATP53MAPTMAPK1
SCHEMBL17865952 0.83 KDM4E (0.48) KDM4ELMNATP53MAPTMAPK1
SCHEMBL17865943 0.79 KDM4E (0.47) KDM4ELMNATP53MAPTMAPK1
SCHEMBL17865941 0.79 NAE1 (0.49) KDM4ELMNATP53MAPTMAPK1
SCHEMBL191796 0.78 NAE1 (0.63) KDM4ELMNATP53MAPTAURKA
SCHEMBL10235267 0.76 NAE1 (0.47) KDM4ELMNATP53MAPTMAPK1
SCHEMBL21283384 0.75 UBA6 (0.46) KDM4ELMNATP53MAPTMAPK1
SCHEMBL16414565 0.72 PRMT5 (0.43)
SCHEMBL22400280 0.70 NAE1 (0.61) AURKARPS6KB1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101379061-A E1 activating enzyme inhibitor MILLENNIUM PHARM INC (US) 2009-03-04 CN disclosed