SCHEMBL27765248

SCHEMBL27765248

CCS(=O)(=O)c1c(-c2ccccc2)cccc1-c1ccc2cccc(C(F)(F)F)c2n1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 7/20 0.40
NR1H3 Q13133 6/20 0.40
PPARG P37231 1/20 0.37
RORC P51449 1/20 0.36
ESR1 P03372 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMO O15229 1/20 0.35
PTGS2 P35354 1/20 0.35
HSD11B1 P28845 1/20 0.34
PARP1 P09874 1/20 0.34
SLC40A1 Q9NP59 1/20 0.34
PTPN1 P18031 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4174099 0.88 PTGS2 (0.41) NR1H2NR1H3ESR1KMOPTGS2
SCHEMBL4164422 0.85 NR1H2 (0.38) NR1H2NR1H3PPARGESR1KMO
SCHEMBL4165443 0.81 NR1H2 (0.44) NR1H2NR1H3RORCESR1CYP1A2
SCHEMBL27765245 0.80 NR1H2 (0.46) NR1H2NR1H3SLC40A1
SCHEMBL28780790 0.79 NR1H2 (0.37) NR1H2NR1H3PPARGRORCESR1
SCHEMBL4164838 0.79 SLC6A2 (0.36) CYP1A2CYP2C19
SCHEMBL27786915 0.79 ESR1 (0.40) NR1H2NR1H3PPARGESR1CYP1A2
SCHEMBL27786978 0.78 KDM4E (0.43) NR1H2NR1H3PPARGRORCESR1
SCHEMBL28780789 0.78 SLC40A1 (0.38) NR1H2NR1H3KMOHSD11B1SLC40A1
SCHEMBL4165744 0.77 PARP1 (0.44) NR1H2NR1H3PPARGRORCCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN claimed
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN disclosed