SCHEMBL4174099

SCHEMBL4174099

CS(=O)(=O)c1c(-c2ccccc2)cccc1-c1ccc2cccc(C(F)(F)F)c2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.41
LMNA P02545 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
SDHB P21912 2/20 0.40
MEN1 O00255 1/20 0.40
S1PR4 O95977 1/20 0.40
TP53 P04637 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
S1PR1 P21453 1/20 0.40
MAPK1 P28482 1/20 0.40
STAT3 P40763 1/20 0.40
STAT1 P42224 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TLR9 Q9NR96 1/20 0.40
NR1H2 P55055 7/20 0.38
NR1H3 Q13133 6/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27765248 0.88 NR1H2 (0.40) PTGS2NR1H2NR1H3ESR1KMO
SCHEMBL4164422 0.87 NR1H2 (0.38) PTGS2NR1H2NR1H3ESR1KMO
SCHEMBL4167348 0.82 NR1H2 (0.41) PTGS2LMNANPSR1SDHBMEN1
SCHEMBL27786915 0.81 ESR1 (0.40) MAPK1HSD17B10NR1H2NR1H3ESR1
SCHEMBL27786940 0.80 NR1H2 (0.42) LMNANPSR1SDHBMEN1S1PR4
SCHEMBL4156275 0.80 PTGS2 (0.39) PTGS2LMNANPSR1SDHBMEN1
SCHEMBL27765196 0.79 PTGS2 (0.64) PTGS2LMNANPSR1MEN1TP53
SCHEMBL4174108 0.79 NR1H3 (0.46) LMNANPSR1SDHBMEN1S1PR4
SCHEMBL27765478 0.78 NR1H2 (0.37) LMNANPSR1SDHBMEN1S1PR4
SCHEMBL28780680 0.78 P2RX7 (0.37) LMNANPSR1SDHBMEN1S1PR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN claimed
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN disclosed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed