SCHEMBL27765461

SCHEMBL27765461

CC(C(=O)C(C)N1CCN(c2ccc(N)nc2)CC1)N1CCN(c2ccc(N)nc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPC6 Q9Y210 3/20 0.44
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
KMT2A Q03164 2/20 0.41
GCK P35557 2/20 0.41
GCKR Q14397 1/20 0.41
HRH3 Q9Y5N1 6/20 0.41
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
F12 P00748 3/20 0.39
CASP6 P55212 1/20 0.38
GFER P55789 1/20 0.38
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL611676 0.83 KDM4E (0.53) TRPC6KDM4EALDH1A1GCKGCKR
SCHEMBL30664050 0.83 KDM4E (0.53) TRPC6KDM4EALDH1A1GCKGCKR
SCHEMBL27563954 0.80 GFER (0.58) KDM4EALDH1A1KMT2AMAPTPKM
SCHEMBL27765462 0.80 TRPC6 (0.39) TRPC6KDM4EALDH1A1GCKGCKR
SCHEMBL27765211 0.79 MAPT (0.60) KDM4EALDH1A1KMT2AMAPTGAA
SCHEMBL29544175 0.78 CASP6 (0.64) TRPC6KMT2AMAPTCASP6GFER
SCHEMBL2450248 0.78 CASP6 (0.64) TRPC6KMT2AMAPTCASP6GFER
SCHEMBL27833098 0.77 HRH3 (0.48) ALDH1A1KMT2AHRH3
SCHEMBL24375241 0.77 GCK (0.39) TRPC6KDM4EALDH1A1GCKGCKR
SCHEMBL29600699 0.76 TRPC6 (0.52) TRPC6ALDH1A1KMT2AGCKGCKR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101594871-B Pyrrolopyrimidine compounds and their uses NOVARTIS AG 2013-06-19 CN disclosed
CN-101594871-A Pyrrolopyrimidine compounds and uses thereof NOVARTIS AG (CH) 2009-12-02 CN disclosed