SCHEMBL27765641

SCHEMBL27765641

Cc1cc2ccc(-c3ccc(O)cc3)cc2[nH]1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 2/20 0.50
FGFR2 P21802 2/20 0.50
FGFR3 P22607 2/20 0.50
ESR1 P03372 8/20 0.48
ESR2 Q92731 6/20 0.48
CDK5 Q00535 3/20 0.48
CDK5R1 Q15078 3/20 0.48
ALOX5 P09917 1/20 0.45
PTGS2 P35354 1/20 0.44
DHODH Q02127 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CDK4 P11802 1/20 0.41
CCND1 P24385 1/20 0.41
HSD17B1 P14061 1/20 0.39
HSD17B2 P37059 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27765605 0.85 PTGS2 (0.59) FGFR1FGFR2FGFR3ESR1ESR2
SCHEMBL30648021 0.84 CA2 (0.50) CDK5CDK5R1MEN1KMT2A
SCHEMBL93623 0.84 CA2 (0.50) CDK5CDK5R1MEN1KMT2A
SCHEMBL13541757 0.83 TNKS2 (0.49) FGFR1ESR1ESR2CDK5CDK5R1
SCHEMBL20615410 0.81 TNKS2 (0.50) FGFR1FGFR2FGFR3PTGS2
SCHEMBL18000095 0.80 PDE3B (0.50)
SCHEMBL28548436 0.79 AXL (0.59) ESR2HSD17B1HSD17B2
SCHEMBL28561888 0.77 MAPT (0.46) PTGS2
SCHEMBL27765642 0.76 ESR2 (0.51) ESR2DHODHMEN1KMT2A
SCHEMBL20494223 0.74 SMAD3 (0.60) FGFR1FGFR2FGFR3ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541801-A Fused heterocyclic derivative and use thereof TAKEDA PHARMACEUTICAL (JP) 2009-09-23 CN disclosed