SCHEMBL27768678

SCHEMBL27768678

O=C(c1csc(-c2ccccc2)n1)c1csc(-c2ccccc2)n1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.70
HDAC8 Q9BY41 1/20 0.70
HDAC6 Q9UBN7 1/20 0.70
TDP1 Q9NUW8 2/20 0.66
HPGDS O60760 2/20 0.60
TLR7 Q9NYK1 1/20 0.60
MAPT P10636 3/20 0.59
ATM Q13315 2/20 0.59
NPSR1 Q6W5P4 2/20 0.59
L3MBTL1 Q9Y468 2/20 0.59
NPY1R P25929 1/20 0.59
NPY2R P49146 1/20 0.59
HPGD P15428 2/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
ALDH1A1 P00352 2/20 0.57
SMN1; SMN2 Q16637 3/20 0.55
KDM4E B2RXH2 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1683594 0.91 HDAC1 (0.64) HDAC1HDAC8HDAC6TDP1HPGDS
SCHEMBL1683722 0.90 TLR7 (0.72) HDAC1HDAC8HDAC6TDP1HPGDS
SCHEMBL352152 0.89 HPGDS (0.73) HDAC1HDAC8HDAC6TDP1HPGDS
Hydrochloric Acid SCHEMBL6821751 0.87 HPGDS (0.71) HDAC1HDAC8HDAC6TDP1HPGDS
SCHEMBL786691 0.85 HDAC1 (0.57) HDAC1HDAC8HDAC6TDP1HPGDS
SCHEMBL1574742 0.85 HDAC1 (0.66) HDAC1HDAC8HDAC6TDP1HPGDS
SCHEMBL168519 0.85 HTR2B (0.66) HDAC1HDAC8HDAC6TDP1HPGDS
SCHEMBL26319518 0.85 ALDH1A1 (0.73) HDAC1HDAC8HDAC6TDP1HPGDS
SCHEMBL168291 0.85 TDP1 (0.67) HDAC1HDAC8HDAC6TDP1HPGDS
SCHEMBL27768683 0.85 HPGD (0.68) HDAC1HDAC8HDAC6TDP1TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102137592-A Compounds for the treatment of cancer UNIV TENNESSEE RES FOUNDATION (US) 2011-07-27 CN claimed
CN-102850324-A Indole compounds MICROBIA INC 2013-01-02 CN disclosed
CN-102137592-A Compounds for the treatment of cancer UNIV TENNESSEE RES FOUNDATION (US) 2011-07-27 CN disclosed
CN-102083839-A Compound (I) ASTRAZENECA AB 2011-06-01 CN disclosed
CN-101563337-A Indole compounds MICROBIA INC (US) 2009-10-21 CN disclosed