SCHEMBL27768752

SCHEMBL27768752

CC(C)(C)OC(=O)N=CCC(CC(=O)O)C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.36
FOLH1 Q04609 2/20 0.34
CTSK P43235 2/20 0.31
CPA1 P15085 2/20 0.30
CPB1 P15086 1/20 0.30
CPA3 P15088 1/20 0.30
CPB2 Q96IY4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27654746 0.84 GAA (0.33) MEN1GAAKMT2ACTSK
SCHEMBL27921297 0.79 MEN1 (0.33) MEN1GAAKMT2ACTSK
SCHEMBL27710328 0.79 MEN1 (0.33) MEN1GAAKMT2ACTSK
SCHEMBL27845696 0.79 MEN1 (0.33) MEN1GAAKMT2ACTSK
SCHEMBL29846523 0.76 CTSK (0.33) CTSK
SCHEMBL27640595 0.73 NOS1 (0.33) CTSK
SCHEMBL25698306 0.70 NPC1 (0.36) KMT2ACTSK
SCHEMBL27274232 0.68 ACLY (0.32)
SCHEMBL28086823 0.68 KMT2A (0.39) MEN1GAAKMT2AFOLH1
SCHEMBL24387451 0.68 CACNA2D1 (0.38) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101611026-A Preparation method of (3R,4R) -N- (4-chlorphenyl) -1- (2, 2-difluoroethyl) -N' - [ 2-fluoro-4- (2-oxo-1 (2H) -pyridyl) phenyl ] -3, 4-pyrrolidine dicarboxamide HOFFMANN LA ROCHE (CH) 2009-12-23 CN disclosed