SCHEMBL2777095

SCHEMBL2777095

CN(CCO)CCCC1CCc2cc(N)ccc2N1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.34
FFAR4 Q5NUL3 1/20 0.32
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
LSS P48449 1/20 0.31
AR P10275 1/20 0.30
ADRA2A P08913 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2776698 0.93 MTNR1A (0.35) MTNR1AFFAR4ESR1ESR2AR
SCHEMBL2778779 0.81 PNMT (0.46) ARADRA2AADRA2BADRA2C
SCHEMBL2778013 0.79 PNMT (0.39) MTNR1AFFAR4ESR1ESR2AR
SCHEMBL2778693 0.77 ACHE (0.41) MTNR1AFFAR4
SCHEMBL15263464 0.74 CA9 (0.41) MTNR1AFFAR4AR
SCHEMBL2777417 0.72 ACHE (0.41) MTNR1AFFAR4LSS
SCHEMBL2781327 0.70 NR1H2 (0.36) MTNR1AFFAR4AR
SCHEMBL2780371 0.70 MTNR1A (0.38) MTNR1AFFAR4AR
SCHEMBL7140193 0.69 MTNR1A (0.34) MTNR1AESR1ESR2
SCHEMBL9394761 0.67 AR (0.40) MTNR1AESR1ESR2AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139886-A1 QUINOLONE AND TETRAHYDROQUINOLINE AND RELATED COMPOUNDS HAVING NOS INHIBITORY ACTIVITY Neuraxon Inc. (CA) 2010-01-06 EP disclosed
WO-2008116308-A1 QUINOLONE AND TETRAHYDROQUINOLINE AND RELATED COMPOUNDS HAVING NOS INHIBITORY ACTIVITY NEURAXON, INC. (CA) 2008-10-02 WO disclosed