SCHEMBL2777758

SCHEMBL2777758

CC(C)[C@H](NC(=O)O)C(=O)N1CCC(C(=O)c2ccc(F)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.59
HSD11B1 P28845 8/20 0.57
CYP2C19 P33261 2/20 0.53
KMT2A Q03164 2/20 0.53
LMNA P02545 1/20 0.53
TSHR P16473 1/20 0.53
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
MGLL Q99685 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2774895 0.84 KMT2A (0.53) CCR1HSD11B1KMT2ALMNATSHR
SCHEMBL2780495 0.80 CCR1 (0.55) CCR1KMT2ALMNATSHR
SCHEMBL2775803 0.80 CCR1 (0.55) CCR1KMT2ALMNATSHR
SCHEMBL2773596 0.80 CCR1 (0.55) CCR1KMT2ALMNATSHR
SCHEMBL2774188 0.79 CCR1 (0.57) CCR1KMT2ALMNATSHR
Hydrochloric Acid SCHEMBL2773460 0.79 HSD11B1 (0.60) HSD11B1CYP2C19LMNAMGLL
Hydrochloric Acid SCHEMBL2773463 0.79 HSD11B1 (0.60) HSD11B1CYP2C19LMNAMGLL
SCHEMBL2774900 0.79 CCR1 (0.55) CCR1HSD11B1CYP2C19KMT2ALMNA
SCHEMBL2775294 0.78 CCR1 (0.53) CCR1KMT2ALMNATSHR
SCHEMBL10291958 0.77 CCR1 (0.89) CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2258697-A1 HYDROXYQUINOXALINECARBOXAMIDE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2010-12-08 EP disclosed