SCHEMBL27778348

SCHEMBL27778348

CCC(C)(C)C(=O)NCc1ccc(C(F)(F)F)nc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 3/20 0.55
TRPV1 Q8NER1 1/20 0.47
NAMPT P43490 2/20 0.46
PTGES O14684 4/20 0.45
KCNQ3 O43525 1/20 0.45
KCNQ2 O43526 1/20 0.45
KCNQ4 P56696 1/20 0.45
KCNQ5 Q9NR82 1/20 0.45
CSF1R P07333 1/20 0.43
GLS O94925 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA14 Q9ULX7 1/20 0.42
KCNH2 Q12809 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP3A5 P20815 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
KDM1A O60341 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19318505 0.87 PTGES (0.55) TRPV1NAMPTPTGESKCNQ3KCNQ2
SCHEMBL4853173 0.82 TRPV1 (0.49) TRPV1NAMPTKCNQ3KCNQ2KCNQ4
SCHEMBL30791579 0.81 TRPV1 (0.51) TRPV1NAMPTKCNQ3KCNQ2KCNQ4
SCHEMBL14306286 0.81 TRPV1 (0.51) TRPV1NAMPTKCNQ3KCNQ2KCNQ4
SCHEMBL22501639 0.80 TRPV1 (0.52) TRPV1NAMPTKCNQ3KCNQ2KCNQ4
SCHEMBL31236179 0.79 TRPV1 (0.51) TRPV1NAMPTKCNQ3KCNQ2KCNQ4
SCHEMBL27799310 0.79 RIPK1 (0.67) RIPK1NAMPT
SCHEMBL10263975 0.78 L3MBTL1 (0.50) TRPV1NAMPTKCNQ3KCNQ2KCNQ4
SCHEMBL14279029 0.78 PTGES (0.56) TRPV1NAMPTPTGESKCNQ3KCNQ2
SCHEMBL2138280 0.76 EPHX2 (0.61) CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101679457-A Piperazine and [1,4] diazepane derivatives as NK antagonists HOFFMANN LA ROCHE 2010-03-24 CN disclosed