SCHEMBL27780484

SCHEMBL27780484

NC(=O)OC(=O)c1ccsc1N

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.62
MEN1 O00255 4/20 0.62
ALDH1A1 P00352 4/20 0.62
MAPT P10636 4/20 0.62
MAPK1 P28482 1/20 0.62
HSD17B10 Q99714 4/20 0.49
USP2 O75604 1/20 0.49
LMNA P02545 1/20 0.49
GLA P06280 1/20 0.49
RAB9A P51151 5/20 0.46
NPC1 O15118 4/20 0.46
PTK2 Q05397 1/20 0.36
MAPK10 P53779 3/20 0.36
POLB P06746 1/20 0.34
TP53 P04637 2/20 0.33
HPGD P15428 2/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
MAPK8 P45983 2/20 0.33
GAA P10253 1/20 0.33
PKM P14618 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL190088 0.78 KMT2A (0.59) KMT2AMEN1ALDH1A1MAPTMAPK1
SCHEMBL164691 0.77
SCHEMBL27854840 0.74 MEN1 (0.71) KMT2AMEN1ALDH1A1MAPTMAPK1
SCHEMBL4144275 0.74 ALDH1A1 (0.53) KMT2AMEN1ALDH1A1MAPTMAPK1
SCHEMBL7799474 0.74 ALDH1A1 (0.53) KMT2AMEN1ALDH1A1MAPTMAPK1
SCHEMBL225275 0.74 ALDH1A1 (0.54) KMT2AMEN1ALDH1A1MAPTMAPK1
SCHEMBL27780712 0.73 KMT2A (0.38) KMT2AMEN1ALDH1A1MAPTMAPK1
SCHEMBL17147852 0.73 ALDH1A1 (0.58) KMT2AMEN1ALDH1A1MAPTMAPK1
SCHEMBL793606 0.73
SCHEMBL28359948 0.72 KMT2A (0.50) KMT2AMEN1ALDH1A1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110759889-B 2-aryl amido substituted thiophene imide ester compound and preparation method and application thereof 中国医学科学院药物研究所 2022-05-20 CN disclosed
CN-110759889-A 2-aryl amido substituted thiophene imide ester compound and preparation method and application thereof 中国医学科学院药物研究所 2020-02-07 CN disclosed
CN-101535276-B 2, 4-diaminopyrimidine fused bicyclic derivatives as ALK and c-MET inhibitors CEPHALON INC 2013-08-28 CN disclosed
CN-101535276-A 2, 4-diaminopyrimidine fused bicyclic derivatives as ALK and c-MET inhibitors CEPHALON INC (US) 2009-09-16 CN disclosed