SCHEMBL27780964

SCHEMBL27780964

O=CC1NCc2ccc(Br)cc21

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PNMT P11086 12/20 0.44
ADRA2A P08913 4/20 0.44
ADRA2B P18089 3/20 0.44
ADRA2C P18825 3/20 0.44
CMA1 P23946 1/20 0.39
AHR P35869 1/20 0.39
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
ASIC3 Q9UHC3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27760113 0.86 PNMT (0.44) PNMTADRA2AADRA2BADRA2CCMA1
SCHEMBL27797441 0.83 HTR2A (0.50) PNMTADRA2AADRA2BADRA2CHTR2A
SCHEMBL27650137 0.79 CHRNB2 (0.35)
SCHEMBL27670223 0.79 DRD2 (0.43) HTR2C
SCHEMBL27923870 0.79 PNMT (0.41) PNMTADRA2AADRA2BADRA2C
SCHEMBL27543455 0.79 CHRNB2 (0.35)
SCHEMBL27650127 0.79 PNMT (0.41) PNMTADRA2AADRA2BADRA2CCMA1
SCHEMBL27884574 0.76 DRD2 (0.33)
SCHEMBL30435099 0.74 CYP2D6 (0.38) ADRA2AADRA2BADRA2C
SCHEMBL3087062 0.74 CYP2D6 (0.38) ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429333-B Synthesis method of gatifloxacin intermediate 江苏法安德医药科技有限公司 2022-03-04 CN disclosed
CN-110938028-B Preparation method of (1R) -5-bromo-2, 3-dihydro-1-methyl-1H-isoindole 南京杰运医药科技有限公司 2022-03-04 CN disclosed
CN-113429333-A Synthesis method of gatifloxacin intermediate 江苏法安德医药科技有限公司 2021-09-24 CN disclosed
CN-110938028-A Preparation method of (1R) -5-bromo-2, 3-dihydro-1-methyl-1H-isoindole 南京杰运医药科技有限公司 2020-03-31 CN disclosed
CN-102858767-B As the aminopyrimidine of SYK inhibitor MERCK SHARP & DOHME CORP. (US) 2015-08-19 CN disclosed
CN-102858767-A Aminopyrimidines as SYK inhibitors MERCK SHARP & DOHME 2013-01-02 CN disclosed
CN-101558067-A 2-methylmorpholine pyrido-, pyrazo- and pyrimido-pyrimidine derivatives as MTOR inhibitors KUDOS PHARM LTD (GB) 2009-10-14 CN disclosed