SCHEMBL27780980

SCHEMBL27780980

CCOC(=O)CC1(O)C(=O)Nc2ccc([N+](=O)[O-])cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
IDO1 P14902 2/20 0.44
MAPT P10636 4/20 0.44
GLO1 Q04760 1/20 0.44
MMP8 P22894 1/20 0.43
AKR1B1 P15121 1/20 0.43
GSK3B P49841 1/20 0.42
KDM4E B2RXH2 1/20 0.42
PGR P06401 1/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
MAPK1 P28482 1/20 0.42
ACHE P22303 1/20 0.41
KMT2A Q03164 1/20 0.41
CACNA1F O60840 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
CACNA1D Q01668 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16377139 0.81 ALDH1A1 (0.54) ALDH1A1CYP3A4CYP2C9CYP2C19IDO1
SCHEMBL27780994 0.80 USP2 (0.55) ALDH1A1CYP2C9CYP2C19IDO1MAPT
SCHEMBL699106 0.80 IDO1 (0.48) ALDH1A1CYP2C9CYP2C19IDO1MAPT
SCHEMBL14609116 0.77 BRD4 (0.40) ALDH1A1CYP3A4CYP2C9CYP2C19IDO1
SCHEMBL14547140 0.75 ALDH1A1 (0.44) ALDH1A1CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL734639 0.75 IDO1 (0.47) ALDH1A1IDO1MAPTLMNA
SCHEMBL18722720 0.73 MMP8 (0.52) ALDH1A1CYP3A4CYP2C9CYP2C19MMP8
SCHEMBL4507525 0.72 AKR1B1 (0.51) ALDH1A1CYP3A4CYP2C9CYP2C19MAPT
SCHEMBL13234058 0.72 ALDH1A1 (0.43) ALDH1A1MAPTGLO1KDM4ELMNA
5-Fluoroisatin SCHEMBL734148 0.72 MAOB (0.41) ALDH1A1IDO1MAPTGSK3BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101516844-B 4-heteroaryl substituted 1-aminocyclohexane-1-and cyclohexene-1-derivatives having activity on opioid receptor systems GRUENENTHAL GMBH 2013-12-11 CN disclosed
CN-101516844-A 4-heteroaryl substituted 1-aminocyclohexane-1-and cyclohexene-1-derivatives having activity on opioid receptor systems GRUENENTHAL GMBH (DE) 2009-08-26 CN disclosed