SCHEMBL2778701

SCHEMBL2778701

CC(O)CCC(C#N)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.48
LMNA P02545 3/20 0.39
TRPA1 O75762 2/20 0.39
CCR1 P32246 1/20 0.39
ADRA2C P18825 2/20 0.38
KDM4E B2RXH2 2/20 0.38
ADRA2A P08913 1/20 0.38
HIF1A Q16665 1/20 0.38
RIPK1 Q13546 1/20 0.38
ALDH1A1 P00352 3/20 0.37
ESR1 P03372 3/20 0.37
ESR2 Q92731 3/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
ALOX5 P09917 1/20 0.37
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37
KMT2A Q03164 1/20 0.37
CHRM2 P08172 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1127660 0.85 TRPA1 (0.42) TSHRLMNATRPA1CCR1ADRA2A
SCHEMBL11865382 0.83 TSHR (0.50) TSHRLMNATRPA1ADRA2CKDM4E
SCHEMBL3432213 0.82 KMT2A (0.44) LMNACCR1KDM4EALDH1A1ESR1
SCHEMBL953748 0.79 TRPA1 (0.43) TSHRLMNATRPA1CCR1ALDH1A1
SCHEMBL988253 0.79 TSHR (0.48) TSHRLMNATRPA1CCR1KDM4E
SCHEMBL27542822 0.76 ALOX5 (0.40) TSHRLMNATRPA1CCR1KDM4E
SCHEMBL27587669 0.76 HRH1 (0.50) LMNAADRA2CKDM4EADRA2AHIF1A
SCHEMBL28981578 0.76 TSHR (0.45) TSHRLMNATRPA1CCR1ALDH1A1
SCHEMBL1445763 0.76 CCR1 (0.42) TSHRLMNATRPA1CCR1KDM4E
SCHEMBL6938022 0.75 HRH1 (0.44) TSHRLMNATRPA1CCR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2266967-A1 Intermediates for the preparation of octahydroquinolizines 55pharma Drug Discovery & Development AG (AT) 2010-12-29 EP disclosed
EP-2266967-A1 Intermediates for the preparation of octahydroquinolizines 55pharma Drug Discovery & Development AG (AT) 2010-12-29 EP disclosed
WO-2010144937-A2 INTERMEDIATES FOR THE PREPARATION OF OCTAHYDROQUINOLIZINES 55PHARMA DRUG DISCOVERY & DEVELOPMENT AG (AT) 2010-12-23 WO disclosed