SCHEMBL27787147

SCHEMBL27787147

NC(=O)C(C(N)=O)S(=O)(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.49
CA1 P00915 4/20 0.47
CA2 P00918 4/20 0.47
CA9 Q16790 2/20 0.47
CA12 O43570 1/20 0.47
MAPT P10636 1/20 0.47
SLC1A3 P43003 1/20 0.47
SLC1A2 P43004 1/20 0.47
SLC1A1 P43005 1/20 0.47
MMP1 P03956 3/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
MMP9 P14780 3/20 0.41
MMP7 P09237 2/20 0.41
MMP2 P08253 2/20 0.41
MMP3 P08254 2/20 0.41
MMP13 P45452 1/20 0.41
PTGS1 P23219 2/20 0.41
PTGS2 P35354 2/20 0.41
GSK3B P49841 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8949440 0.77 SLC1A3 (0.49) KIF11CA1CA2CA9CA12
SCHEMBL4225010 0.76 KIF11 (0.53) KIF11CA1CA2CA9CA12
SCHEMBL8619633 0.75 SLC1A2 (0.61) KIF11CA1CA2CA9CA12
SCHEMBL3151057 0.74 KIF11 (0.59) KIF11CA1CA2CA9CA12
SCHEMBL1464399 0.74 MMP1 (0.54) KIF11CA1CA2CA9CA12
SCHEMBL10157181 0.73 CA1 (0.53) KIF11CA1CA2CA9CA12
SCHEMBL28200284 0.72 CES2 (0.50) KIF11CA1CA2CA9CES2
SCHEMBL1465778 0.71 MMP1 (0.55) KIF11CA1CA2CA9CA12
SCHEMBL13833092 0.70 KIF11 (0.47) KIF11CA1CA2CA9CA12
SCHEMBL230582 0.70 KIF11 (0.55) KIF11CA1CA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101784520-B Novel malonic acid sulfonamide derivative and pharmaceutical use thereof MITSUBISHI TANABE PHARMA CORP 2014-07-02 CN disclosed
CN-101784520-A Novel malonic acid sulfonamide derivative and pharmaceutical use thereof MITSUBISHI TANABE PHARMA CORP 2010-07-21 CN disclosed