SCHEMBL27787706

SCHEMBL27787706

CC(C)(C)C(=O)ON1CCN(CC(=O)c2ccc(F)cc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
TSHR P16473 3/20 0.51
KDM4E B2RXH2 2/20 0.51
HTT P42858 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
HTR2A P28223 10/20 0.49
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
CYP2C19 P33261 2/20 0.48
GAA P10253 2/20 0.48
PKM P14618 1/20 0.48
ALOX15 P16050 1/20 0.48
HTR2C P28335 6/20 0.48
MAPT P10636 1/20 0.48
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
USP2 O75604 1/20 0.46
HPGD P15428 1/20 0.46
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28060545 0.80 POLB (0.51) ALDH1A1HTTSMN1; SMN2MEN1KMT2A
SCHEMBL17180311 0.79 HTR2A (0.57) ALDH1A1TSHRKDM4EHTTSMN1; SMN2
SCHEMBL27787732 0.79 HTR2A (0.49) HTR2AHTR2CKCNH2
SCHEMBL9660142 0.77 TSHR (0.68) ALDH1A1TSHRKDM4EHTTSMN1; SMN2
SCHEMBL27731418 0.77 LTA4H (0.52) ALDH1A1KDM4EHTTMEN1KMT2A
SCHEMBL27758338 0.76 HSD11B1 (0.57) ALDH1A1KDM4ESMN1; SMN2HTR2AGAA
SCHEMBL9871356 0.75 ALDH1A1 (0.61) ALDH1A1TSHRKDM4EHTTSMN1; SMN2
SCHEMBL27758590 0.75 KMT2A (0.37) ALDH1A1SMN1; SMN2CYP2D6MEN1KMT2A
SCHEMBL7462619 0.75 ALDH1A1 (0.71) ALDH1A1TSHRKDM4EHTTSMN1; SMN2
Hydrochloric Acid SCHEMBL10369554 0.74 ALDH1A1 (0.60) ALDH1A1TSHRKDM4EHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102838546-B Pyrazole derivatives as modulators of 5-ht2a serotonin receptor useful for treatment of disorders related thereto ARENA PHARM INC 2015-07-15 CN disclosed
CN-102838546-A Pyrazole derivatives as modulators of 5-ht2a serotonin receptor useful for treatment of disorders related thereto ARENA PHARM INC 2012-12-26 CN disclosed
CN-101611013-B As 5-HT2APyrazole derivatives of serotonin receptor modulators for the treatment of disorders related thereto ARENA PHARM INC 2012-09-05 CN disclosed
CN-101611013-A As 5-HT2APyrazole derivatives of serotonin receptor modulators for the treatment of disorders related thereto ARENA PHARM INC (US) 2009-12-23 CN disclosed