SCHEMBL27794864

SCHEMBL27794864

O=C(O)c1cnc(Cc2ccccc2F)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 1/20 0.50
RARA P10276 1/20 0.45
RARB P10826 1/20 0.45
RARG P13631 1/20 0.45
GCK P35557 1/20 0.45
ALKBH1 Q13686 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
ATM Q13315 1/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
KDM5A P29375 3/20 0.43
KDM5B Q9UGL1 3/20 0.43
KDM4A O75164 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
PTPN1 P18031 1/20 0.42
BRS3 P32247 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL456951 0.78 LDHA (0.46) VNN1KDM5AKDM5BKDM4CMEN1
SCHEMBL9485705 0.75 NPC1 (0.49) KDM4EALDH1A1HPGDHSD17B10HTR2C
SCHEMBL24230227 0.75 TSHR (0.67) ALDH1A1HPGDATMPTPN1LPAR1
SCHEMBL15737161 0.73 NR4A2 (0.49) VNN1ALKBH1HTR2CHTR2BKDM5A
SCHEMBL11828345 0.73 RXRA (0.53) KDM4EATMKDM5AKDM5BKDM4A
SCHEMBL4677195 0.73 GCK (0.59) VNN1RARARARBRARGGCK
SCHEMBL4636142 0.73 DHODH (0.48) VNN1HPGDKDM5AKDM5BKDM4C
SCHEMBL3226195 0.72 NR4A2 (0.54) ALKBH1HTR2CHTR2BKDM5AKDM5B
SCHEMBL20894099 0.71 NPC1 (0.45) VNN1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL29631019 0.71 NPC1 (0.45) VNN1KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101646656-A Pyrimidine hydrazide compounds as the PGDS inhibitor SANOFI AVENTIS FR 2010-02-10 CN claimed
CN-101646656-B Pyrimidine hydrazide compounds as PGDS inhibitors SANOFI AVENTIS SPA 2013-08-14 CN disclosed
CN-101646656-A Pyrimidine hydrazide compounds as the PGDS inhibitor SANOFI AVENTIS FR 2010-02-10 CN disclosed