SCHEMBL27794865

SCHEMBL27794865

COc1ccc(Oc2ccccc2)nc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 3/20 0.57
KDM4E B2RXH2 4/20 0.54
ALDH1A1 P00352 2/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
BRCA1 P38398 1/20 0.54
HBB P68871 1/20 0.54
HSD17B10 Q99714 1/20 0.54
HTT P42858 2/20 0.53
RAB9A P51151 2/20 0.53
NPC1 O15118 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
RXFP1 Q9HBX9 1/20 0.53
HAO1 Q9UJM8 2/20 0.49
CA4 P22748 1/20 0.48
LMNA P02545 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
OXTR P30559 1/20 0.44
AVPR1A P37288 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28760544 0.86 LTA4H (0.52) LTA4HKDM4EALDH1A1MEN1KMT2A
SCHEMBL27961825 0.83 HAO1 (0.51) KDM4EALDH1A1MEN1KMT2ABRCA1
SCHEMBL177968 0.83 KDM4E (0.61) KDM4EALDH1A1MEN1KMT2ABRCA1
SCHEMBL16838784 0.83 HAO1 (0.47) KDM4EALDH1A1MEN1KMT2ABRCA1
SCHEMBL21525575 0.81 CA1 (0.59) KDM4EHTTRAB9ANPC1LMNA
SCHEMBL3816388 0.79 NNMT (0.48) KDM4EALDH1A1MEN1KMT2ABRCA1
SCHEMBL29525223 0.79 NNMT (0.48) KDM4EALDH1A1MEN1KMT2ABRCA1
SCHEMBL16838765 0.79 LMNA (0.59) KDM4EHTTRAB9ANPSR1LMNA
SCHEMBL27368615 0.79 OPRM1 (0.46) KDM4EALDH1A1MEN1KMT2ABRCA1
SCHEMBL8306130 0.78 KDM4E (0.53) LTA4HKDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103201261-A Lactam derivatives as orexin receptor antagonists ACTELION PHARMACEUTICALS LTD 2013-07-10 CN disclosed
CN-101842357-A Substituted pyrazole derivatives TAKEDA PHARMACEUTICAL 2010-09-22 CN disclosed