SCHEMBL27801909

SCHEMBL27801909

CCc1nocc1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.44
HSP90AA1 P07900 1/20 0.42
PTGS1 P23219 1/20 0.40
DHFR P00374 1/20 0.39
HEXA P06865 1/20 0.39
HEXB P07686 1/20 0.39
ADORA3 P0DMS8 2/20 0.38
NOTUM Q6P988 5/20 0.37
GCGR P47871 1/20 0.36
TP53 P04637 2/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GPR55 Q9Y2T6 1/20 0.34
TDO2 P48775 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28763009 0.85 PTGS2 (0.42) PTGS2HSP90AA1PTGS1ADORA3NOTUM
SCHEMBL5668350 0.82 HSP90AA1 (0.47) PTGS2HSP90AA1ADORA3NOTUMRAB9A
SCHEMBL19465377 0.81 SMN1; SMN2 (0.41) DHFRHEXAHEXBNOTUMTP53
SCHEMBL6630456 0.81 PTGS2 (0.44) PTGS2HSP90AA1ADORA3NOTUMTP53
SCHEMBL27425761 0.79 RAB9A (0.42) PTGS2HSP90AA1ADORA3NOTUMNPC1
SCHEMBL4454083 0.77 CASP3 (0.39) HSP90AA1TP53NPC1LMNARAB9A
SCHEMBL6630766 0.74 PTGS2 (0.47) PTGS2HSP90AA1PTGS1NOTUMTP53
SCHEMBL6632000 0.72 MAPT (0.52) ADORA3LMNASMN1; SMN2ALDH1A1
SCHEMBL1797330 0.71 PTGS2 (0.67) PTGS2HSP90AA1PTGS1NOTUMTP53
SCHEMBL10983313 0.70 KDM4E (0.46) NPC1LMNARAB9ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101715451-A Novel pyridopyrazine derivatives, process for their preparation and their use AETERNA ZENTARIS GMBH 2010-05-26 CN claimed
CN-101715451-B Novel pyridopyrazine derivatives, process for their preparation and their use AETERNA ZENTARIS GMBH 2013-07-31 CN disclosed
CN-101715451-A Novel pyridopyrazine derivatives, process for their preparation and their use AETERNA ZENTARIS GMBH 2010-05-26 CN disclosed