SCHEMBL27806830

SCHEMBL27806830

FC(F)(F)c1cc(CP(Cl)(c2ccccc2)(c2ccccc2)c2ccccc2)ccc1OCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RXRA P19793 3/20 0.46
RXRB P28702 3/20 0.46
RXRG P48443 3/20 0.46
MRGPRX4 Q96LA9 8/20 0.46
S1PR1 P21453 4/20 0.41
CTSS P25774 1/20 0.40
HTR2C P28335 1/20 0.39
SLC6A4 P31645 1/20 0.39
HTR2B P41595 1/20 0.39
PTGER1 P34995 1/20 0.36
S1PR4 O95977 1/20 0.36
S1PR5 Q9H228 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL79415 0.81 RXRA (0.52) RXRARXRBRXRGMRGPRX4S1PR1
SCHEMBL79041 0.78 RXRA (0.56) RXRARXRBRXRGMRGPRX4S1PR1
SCHEMBL18924486 0.76 RXRA (0.50) RXRARXRBRXRGMRGPRX4S1PR1
SCHEMBL6812974 0.76 CYP4F2 (0.54) RXRARXRBRXRGMRGPRX4S1PR1
SCHEMBL20756090 0.75 RXRA (0.54) RXRARXRBRXRGMRGPRX4CTSS
SCHEMBL86405 0.75 RXRA (0.49) RXRARXRBRXRGMRGPRX4S1PR1
SCHEMBL656838 0.74 MRGPRX4 (0.50) RXRARXRBRXRGMRGPRX4S1PR1
SCHEMBL5388117 0.74 RXRA (0.60) RXRARXRBRXRGMRGPRX4S1PR1
SCHEMBL14453588 0.74 MRGPRX4 (0.50) RXRARXRBRXRGMRGPRX4S1PR1
SCHEMBL3726426 0.74 PTGER1 (0.54) RXRARXRBRXRGMRGPRX4SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101730677-B Amine compound and pharmaceutical use thereof MITSUBISHI TANABE PHARMA CORP 2014-07-16 CN disclosed
CN-101730677-A Amine compound and pharmaceutical use thereof MITSUBISHI TANABE PHARMA CORP 2010-06-09 CN disclosed