SCHEMBL27807883

SCHEMBL27807883

O=C1N(c2ccccc2)C(C2(C(=O)O)C=CC=C(c3ccccc3)C2)CN1S(=O)(=O)c1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
CTSG P08311 3/20 0.33
CMA1 P23946 3/20 0.33
MCL1 Q07820 2/20 0.33
PKM P14618 3/20 0.32
MMP2 P08253 2/20 0.32
AKR1C3 P42330 2/20 0.31
AKR1C1 Q04828 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MMP9 P14780 1/20 0.30
PARL Q9H300 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27807878 0.83 CYP3A4 (0.35) CYP2D6CYP3A4CYP2C9CYP2C19CTSG
SCHEMBL27807885 0.78 CTSG (0.33) CYP2D6CTSGCMA1MCL1PKM
SCHEMBL27807880 0.74 PKM (0.30) CYP2C9PKMMMP2
SCHEMBL27807884 0.67 MCL1 (0.30) MCL1
SCHEMBL1348740 0.67 CMA1 (0.45) CTSGCMA1MCL1PKMAKR1C3
SCHEMBL28787377 0.67 PKM (0.37) CYP3A4CYP2C9CYP2C19CTSGCMA1
SCHEMBL1348640 0.64 CMA1 (0.44) CTSGCMA1MCL1AKR1C3AKR1C1
SCHEMBL1348608 0.64 MCL1 (0.43) CTSGCMA1MCL1PKMAKR1C3
SCHEMBL1348509 0.63 PKM (0.37) CTSGCMA1MCL1PKMMMP2
SCHEMBL27807891 0.63 ALDH1A1 (0.38) CYP3A4CYP2C9CYP2C19PKMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102056902-B Imidazolidine derivatives HOFFMANN LA ROCHE 2013-08-07 CN claimed
CN-102056902-A Imidazolidine derivatives HOFFMANN LA ROCHE 2011-05-11 CN claimed
CN-102056902-B Imidazolidine derivatives HOFFMANN LA ROCHE 2013-08-07 CN disclosed
CN-102056902-A Imidazolidine derivatives HOFFMANN LA ROCHE 2011-05-11 CN disclosed