SCHEMBL28787377

SCHEMBL28787377

N#CC1(C2CN(S(=O)(=O)c3ccccc3)CC(=O)N2c2ccccc2)C=CC=C(c2ccccc2)C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.37
ALDH1A1 P00352 5/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
CTSG P08311 3/20 0.32
CMA1 P23946 3/20 0.32
TSHR P16473 2/20 0.32
USP2 O75604 4/20 0.31
HSD17B10 Q99714 3/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
HPGD P15428 1/20 0.31
MAPK1 P28482 1/20 0.31
HIF1A Q16665 1/20 0.31
POLB P06746 1/20 0.31
MCL1 Q07820 1/20 0.31
PAX8 Q06710 1/20 0.31
CYP1A2 P05177 3/20 0.31
CYP3A4 P08684 3/20 0.31
CYP2C9 P11712 2/20 0.31
CYP2C19 P33261 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27807878 0.67 CYP3A4 (0.35) PKMALDH1A1CTSGCMA1TSHR
SCHEMBL27807891 0.67 ALDH1A1 (0.38) PKMALDH1A1MEN1KMT2ATSHR
SCHEMBL27807883 0.67 CYP2D6 (0.34) PKMALDH1A1CTSGCMA1MCL1
SCHEMBL1349414 0.65 CTSG (0.47) PKMALDH1A1KMT2ACTSGCMA1
SCHEMBL27828349 0.63 LMNA (0.47) PKMALDH1A1MEN1KMT2ATSHR
SCHEMBL1349030 0.61 NR1H2 (0.41) PKMALDH1A1KMT2AUSP2HSD17B10
SCHEMBL1347358 0.59 MMP2 (0.44) PKMALDH1A1MEN1KMT2ACTSG
SCHEMBL27771620 0.59
SCHEMBL5449733 0.58 PKM (0.54) PKMALDH1A1MEN1KMT2ACTSG
SCHEMBL27878415 0.57

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102056902-B Imidazolidine derivatives HOFFMANN LA ROCHE 2013-08-07 CN disclosed
CN-102056902-A Imidazolidine derivatives HOFFMANN LA ROCHE 2011-05-11 CN disclosed