SCHEMBL4331617

SCHEMBL4331617

[c]1cccc(CCc2cccc(N3CCOCC3)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGXT P21549 2/20 0.55
LMNA P02545 1/20 0.44
KMO O15229 1/20 0.43
AOC3 Q16853 2/20 0.42
SIGMAR1 Q99720 4/20 0.41
TMEM97 Q5BJF2 3/20 0.41
ADRA2A P08913 2/20 0.41
ADRA2B P18089 2/20 0.41
ADRA2C P18825 1/20 0.41
PRMT6 Q96LA8 1/20 0.40
L3MBTL3 Q96JM7 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PLOD2 O00469 2/20 0.39
PLOD3 O60568 2/20 0.39
PLOD1 Q02809 2/20 0.39
DRD4 P21917 1/20 0.39
HRH1 P35367 1/20 0.39
HTR2B P41595 1/20 0.39
KLKB1 P03952 1/20 0.39
KLK1 P06870 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4340373 0.87 MAPT (0.45) AGXTLMNASIGMAR1TMEM97ADRA2A
SCHEMBL4328642 0.87 PRMT6 (0.54) AGXTSIGMAR1PRMT6L3MBTL3L3MBTL1
SCHEMBL4337043 0.83 HTR7 (0.50) SIGMAR1HTR2B
SCHEMBL3141768 0.81 AGXT (0.48) AGXTLMNAKMO
SCHEMBL27809061 0.81 NCF1 (0.58) SIGMAR1PRMT6
SCHEMBL159425 0.78 LMNA (0.59) AGXTLMNAKMO
SCHEMBL27425605 0.78 MAPT (0.44) AGXTLMNASIGMAR1TMEM97ADRA2A
SCHEMBL27829456 0.78 RORC (0.46) AOC3
SCHEMBL13725027 0.78 AGXT (0.66) AGXTLMNAKMOAOC3SIGMAR1
SCHEMBL8189516 0.78 AGXT (0.61) AGXTLMNAKMOAOC3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009145360-A1 BENZENE OR THIOPHENE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-TECH UENO, LTD. (JP) 2009-12-03 WO disclosed