SCHEMBL27809382

SCHEMBL27809382

O=C(O)c1cccc2c1C=CNC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.42
ALDH1A1 P00352 3/20 0.39
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 2/20 0.38
TSHR P16473 1/20 0.35
NR4A1 P22736 1/20 0.35
NR4A2 P43354 1/20 0.35
NR4A3 Q92570 1/20 0.35
KEAP1 Q14145 1/20 0.35
AURKA O14965 1/20 0.35
KDM4E B2RXH2 2/20 0.34
HPGD P15428 2/20 0.34
NAPRT Q6XQN6 2/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
HMGB1 P09429 1/20 0.34
CA4 P22748 1/20 0.34
CA6 P23280 1/20 0.34
CA7 P43166 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4442482 0.85 AURKA (0.47) PARP1ALDH1A1HSD17B10TSHRAURKA
SCHEMBL36891321 0.73 ALDH1A1 (0.43) ALDH1A1ALOX15HSD17B10TSHRNR4A1
SCHEMBL286794 0.73 ALDH1A1 (0.43) ALDH1A1ALOX15HSD17B10TSHRNR4A1
SCHEMBL4202677 0.72 PARP1 (0.42) PARP1ALDH1A1ALOX15HSD17B10TSHR
SCHEMBL16621278 0.71 PARP1 (0.47) PARP1
SCHEMBL5753321 0.70 ALDH1A1 (0.40) PARP1ALDH1A1ALOX15HSD17B10TSHR
SCHEMBL8980518 0.70 PARP1 (0.43) PARP1
SCHEMBL6201130 0.69 ALDH1A1 (0.39) ALDH1A1ALOX15HSD17B10TSHRNR4A1
SCHEMBL20120194 0.69 TDP1 (0.42) PARP1ALDH1A1ALOX15HSD17B10TSHR
Oxalic Acid SCHEMBL21489558 0.68 PARP1 (0.75) PARP1ALDH1A1TSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101790518-A Derivatives of 1-oxo-1, 2-dihydroisoquinoline-5-carboxamides and of 4-oxo-3, 4-dihydroquinazoline-8-carboxamides, preparation thereof and therapeutic use thereof SANOFI AVENTIS 2010-07-28 CN disclosed