SCHEMBL27809403

SCHEMBL27809403

O=C(O)c1nocc1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 1/20 0.46
MAP4K4 O95819 1/20 0.43
PSEN1 P49768 1/20 0.42
PSEN2 P49810 1/20 0.42
APH1B Q8WW43 1/20 0.42
NCSTN Q92542 1/20 0.42
APH1A Q96BI3 1/20 0.42
PSENEN Q9NZ42 1/20 0.42
APP P05067 2/20 0.41
SRD5A2 P31213 1/20 0.41
BACE1 P56817 1/20 0.40
IKBKB O14920 1/20 0.40
TRPV1 Q8NER1 2/20 0.40
NPC1 O15118 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SLC22A12 Q96S37 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27809428 0.82 MAPK14 (0.49) MAP4K4
SCHEMBL27787513 0.81 AURKA (0.45) TRPV1CYP2C9AKR1C2
SCHEMBL4075531 0.80 PTPN1 (0.47) LMNASMN1; SMN2
SCHEMBL27809418 0.79 KIF11 (0.46) TRPV1KIF11
SCHEMBL12466534 0.75 KMO (0.43) LMNASLC22A12AKR1C3AKR1C2CES2
SCHEMBL28268214 0.72 KLRK1 (0.50) CYP2C8MAP4K4BACE1TRPV1
SCHEMBL27809437 0.72 KMO (0.48) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1686231 0.72 TRPV1 (0.61) TRPV1
SCHEMBL27787507 0.72 KMO (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL17288815 0.71 ALDH1A1 (0.43) SRD5A2RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101796036-A 5-Phenylisoxazole-3-carboxamide derivatives as TRPV1 modulators ORGANON NV 2010-08-04 CN disclosed