SCHEMBL12466534

SCHEMBL12466534

O=C(O)c1nocc1-c1ccc(F)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.43
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
IDO1 P14902 1/20 0.39
KDM5A P29375 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
KDM5B Q9UGL1 1/20 0.39
SLC22A12 Q96S37 1/20 0.39
DUSP3 P51452 1/20 0.38
XDH P47989 1/20 0.37
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
KDM4E B2RXH2 2/20 0.35
LMNA P02545 2/20 0.35
HSD17B10 Q99714 2/20 0.35
ACMSD Q8TDX5 2/20 0.35
GRK6 P43250 1/20 0.35
HDAC1 Q13547 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27787507 0.87 KMO (0.47) KMOAKR1C3AKR1C2KDM4CDUSP3
SCHEMBL27809418 0.84 KIF11 (0.46)
SCHEMBL27809428 0.82 MAPK14 (0.49) KMT2A
SCHEMBL27809437 0.78 KMO (0.48) KMOAKR1C3AKR1C2
SCHEMBL4658590 0.77 PIN1 (0.48) KMODUSP3
SCHEMBL4398019 0.77 ALDH1A1 (0.45) DUSP3MAPTKDM4ELMNAHSD17B10
SCHEMBL4075531 0.76 PTPN1 (0.47) DUSP3MAPTKDM4ELMNAALDH1A1
SCHEMBL3228354 0.76 ALDH1A1 (0.39) MAPTKDM4EHSD17B10MEN1USP2
SCHEMBL27809403 0.75 CYP2C8 (0.46) AKR1C3AKR1C2SLC22A12LMNACES2
SCHEMBL4081921 0.75 KMO (0.43) KMOAKR1C3AKR1C2IDO1KDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012103113-A1 PYRAZINE AND IMIDAZOLIDINE DERIVATIVES AND THEIR USES TO TREAT HEPATITIS C GILEAD PHARMASSET, LLC (US) 2012-08-02 WO disclosed