SCHEMBL27823720

SCHEMBL27823720

CCCCc1c(C#N)c2cc(-c3ccc[nH]c3=O)ccc2n1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 6/20 0.40
WDR77 Q9BQA1 6/20 0.40
ALDH1A1 P00352 9/20 0.38
GAA P10253 3/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
TSHR P16473 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
NPC1 O15118 1/20 0.38
GLA P06280 1/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
KDM4E B2RXH2 6/20 0.36
LMNA P02545 2/20 0.36
CYP1A2 P05177 2/20 0.36
HPGD P15428 2/20 0.36
TP53 P04637 1/20 0.36
HIF1A Q16665 1/20 0.36
METAP2 P50579 1/20 0.36
HSD17B10 Q99714 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1971791 0.71 IMPDH2 (0.47) PRMT5WDR77ALDH1A1KDM4ECYP1A2
SCHEMBL27831895 0.68 IGLV6-57 (0.41) ALDH1A1GAAKDM4EMEN1KMT2A
SCHEMBL16518824 0.65 KDM4E (0.41) ALDH1A1GAAL3MBTL1NPC1RAB9A
SCHEMBL15536272 0.62 MCL1 (0.52) NPC1
SCHEMBL15334010 0.62 TRPA1 (0.56) ALDH1A1KDM4ECYP1A2HPGD
SCHEMBL1971648 0.62 KDM4E (0.46) ALDH1A1KDM4ECYP1A2HPGDKMT2A
SCHEMBL3821760 0.62 ALDH1A1 (0.41) ALDH1A1GAAGLARAB9AKDM4E
SCHEMBL27811660 0.61 CNR1 (0.37) ALDH1A1GAAKDM4EKMT2A
SCHEMBL16456343 0.59 TNKS (0.41) ALDH1A1GAAL3MBTL1NPC1MAPK1
SCHEMBL10692239 0.59 DAO (0.41) ALDH1A1GAAL3MBTL1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102164909-A Pyrine or pyrazine derivatives for treating HCV HOFFMANN LA ROCHE 2011-08-24 CN claimed