SCHEMBL27856412

SCHEMBL27856412

COC(=O)c1ccc2ccccc2n1.O=[N+]([O-])c1ccc2c(c1)NCC2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.52
KDM4E B2RXH2 3/20 0.52
GAA P10253 2/20 0.52
MAPT P10636 4/20 0.52
POLB P06746 1/20 0.44
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
RECQL P46063 1/20 0.41
HTT P42858 2/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
NPC1 O15118 1/20 0.37
MAPK1 P28482 1/20 0.37
HPGD P15428 1/20 0.37
SLC6A4 P31645 1/20 0.36
F2 P00734 1/20 0.36
PLAU P00749 1/20 0.36
KLKB1 P03952 1/20 0.36
ELANE P08246 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL27721275 0.79 ALDH1A1 (0.45) ALDH1A1KDM4EGAAMAPTKMT2A
SCHEMBL30663244 0.77 ALDH1A1 (0.54) ALDH1A1KDM4EGAAMAPTPOLB
SCHEMBL6965338 0.76 ALDH1A1 (0.53) ALDH1A1KDM4EGAAMAPTPOLB
SCHEMBL31378863 0.74 PNMT (0.58) ALDH1A1MAPTKMT2AMEN1RAB9A
SCHEMBL427407 0.74 PNMT (0.58) ALDH1A1MAPTKMT2AMEN1RAB9A
Quinoline SCHEMBL28039586 0.74 ALDH1A1 (0.36) ALDH1A1KDM4EGAAMAPTKMT2A
SCHEMBL30208641 0.73 MGAM (0.61) ALDH1A1KDM4EGAAMAPTKMT2A
SCHEMBL725183 0.73 MGAM (0.61) ALDH1A1KDM4EGAAMAPTKMT2A
Hydrochloric Acid SCHEMBL16793838 0.71 MGAM (0.59) ALDH1A1KDM4EGAAMAPTKMT2A
Hydrochloric Acid SCHEMBL30615167 0.71 MGAM (0.59) ALDH1A1KDM4EGAAMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108727407-A Novel benzodiazepine * derivatives 伊缪诺金公司 2018-11-02 CN disclosed
CN-105198908-A Novel benzodiazepine derivatives IMMUNOGEN INC 2015-12-30 CN disclosed
CN-105175434-A NOVEL BENZODIAZEPINE DERIVATIVES IMMUNOGEN INC 2015-12-23 CN disclosed
CN-102365021-B Novel benzodiazepine derivatives IMMUNOGEN INC 2015-07-15 CN disclosed
CN-102365021-A Novel benzodiazepine derivatives IMMUNOGEN INC 2012-02-29 CN disclosed