SCHEMBL27856416

SCHEMBL27856416

O=C(O)NN[C@@H]1CCc2ccc(Br)cc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
ACHE P22303 3/20 0.39
PTGDR Q13258 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
LMNA P02545 1/20 0.37
KMT2A Q03164 1/20 0.37
IDO1 P14902 2/20 0.37
FAAH O00519 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
XIAP P98170 1/20 0.36
SRD5A1 P18405 1/20 0.36
SRD5A2 P31213 1/20 0.36
CTSS P25774 1/20 0.35
CAMK2A Q9UQM7 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27838566 1.00 MAOA (0.40) MAOAMAOBACHEPTGDRPTGDR2
SCHEMBL484798 0.86 LMNA (0.44) MAOAMAOBACHEPTGDRPTGDR2
SCHEMBL19521080 0.78 KMT2A (0.54) LMNAKMT2ACTSS
SCHEMBL28300302 0.78 PDPK1 (0.56) MAOAMAOBACHEKMT2AEPHX2
SCHEMBL28224650 0.78 PDPK1 (0.56) MAOAMAOBACHEKMT2AEPHX2
SCHEMBL30985322 0.76 PDPK1 (0.58) MAOAMAOBACHEHTR2AHTR2C
SCHEMBL805451 0.76 HTR2A (0.46) MAOAMAOBACHEHTR2AHTR2C
SCHEMBL15447552 0.76 PDPK1 (0.58) MAOAMAOBACHEHTR2AHTR2C
SCHEMBL6497708 0.76 PDPK1 (0.58) MAOAMAOBACHEHTR2AHTR2C
SCHEMBL10469026 0.74 FABP4 (0.43) PTGDRPTGDR2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103097354-A Substituted benzamide compounds GRUENENTHAL CHEMIE 2013-05-08 CN disclosed
CN-102365276-A Substituted spiro-amide compounds GRUENENTHAL GMBH 2012-02-29 CN disclosed