SCHEMBL27859136

SCHEMBL27859136

Cc1cc(F)c(C(C)C=O)cc1[N+](=O)[O-]

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
MAPT P10636 3/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TSHR P16473 4/20 0.37
CYP3A4 P08684 2/20 0.37
RECQL P46063 1/20 0.37
TDP1 Q9NUW8 2/20 0.35
ATM Q13315 1/20 0.35
HIF1A Q16665 1/20 0.34
HSD17B10 Q99714 1/20 0.33
GAA P10253 1/20 0.33
CYP1A2 P05177 1/20 0.33
HTT P42858 1/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GPR35 Q9HC97 2/20 0.33
ESPL1 Q14674 1/20 0.33
VCAM1 P19320 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27859137 0.78 TSHR (0.41) ALDH1A1MAPTSMN1; SMN2TSHRCYP3A4
SCHEMBL29525219 0.75 ALDH1A1 (0.53) ALDH1A1MAPTSMN1; SMN2TSHRCYP3A4
SCHEMBL440478 0.75 ALDH1A1 (0.53) ALDH1A1MAPTSMN1; SMN2TSHRCYP3A4
SCHEMBL31361810 0.74 ALDH1A1 (0.41) ALDH1A1MAPTSMN1; SMN2TSHRCYP3A4
SCHEMBL2471756 0.74 ALDH1A1 (0.47) ALDH1A1MAPTSMN1; SMN2TSHRCYP3A4
SCHEMBL397387 0.74 ATM (0.50) ALDH1A1MAPTSMN1; SMN2TSHRCYP3A4
SCHEMBL18216945 0.73 ALDH1A1 (0.45) ALDH1A1MAPTSMN1; SMN2TSHRCYP3A4
SCHEMBL27841693 0.73 POLB (0.39) ALDH1A1TSHRCYP3A4HIF1AHSD17B10
SCHEMBL15927701 0.73 TDP1 (0.43) ALDH1A1MAPTSMN1; SMN2TSHRCYP3A4
SCHEMBL27781739 0.73 ATM (0.51) ALDH1A1MAPTSMN1; SMN2TSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102471284-A Dihydropyrimidone amides as P2X7 modulators HOFFMANN LA ROCHE 2012-05-23 CN disclosed
CN-102264722-A Dihydropyridone amides as p2x7 modulators 2011-11-30 CN disclosed