SCHEMBL2786321

SCHEMBL2786321

O=C(NSc1ccc(F)cc1)Nc1noc2cc(Cl)ccc12

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 5/20 0.44
SMN1; SMN2 Q16637 5/20 0.44
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
KCNJ6 P48051 1/20 0.39
KCNJ3 P48549 1/20 0.39
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38
HTR3A P46098 3/20 0.37
CHRNA7 P36544 2/20 0.37
HSD17B10 Q99714 1/20 0.34
GRIK1 P39086 1/20 0.34
KCNMA1 Q12791 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2787441 0.86 TP53 (0.47) TP53SMN1; SMN2ALOX15TSHRKCNJ6
SCHEMBL2785764 0.86 ABCC9 (0.45) TP53SMN1; SMN2ALOX15TSHRKCNJ6
SCHEMBL2787195 0.83 TP53 (0.63) TP53SMN1; SMN2ALOX15TSHRKCNJ6
SCHEMBL2787058 0.82 TP53 (0.46) TP53SMN1; SMN2ALOX15TSHRKCNJ6
SCHEMBL2785392 0.79 MAPT (0.42) TP53SMN1; SMN2ALOX15TSHRKCNJ6
SCHEMBL2786470 0.75 HTR3A (0.44) TP53SMN1; SMN2ALOX15TSHRKCNJ6
SCHEMBL2768955 0.74 MAOB (0.52) SMN1; SMN2ALDH1A1KMT2AHTR3ACHRNA7
SCHEMBL2787333 0.73 SMN1; SMN2 (0.45) TP53SMN1; SMN2ALOX15ALDH1A1KMT2A
SCHEMBL2785316 0.73 TP53 (0.52) TP53SMN1; SMN2ALOX15TSHRKCNJ6
SCHEMBL2439515 0.72 TP53 (0.48) TP53SMN1; SMN2ALOX15TSHRKCNJ6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881967-B1 SUBSTITUTED BENZO(D)ISOXAZOL-3-YL AMINE COMPOUNDS AS ANALGESICS GRUENENTHAL GMBH (DE) 2010-04-28 EP claimed