SCHEMBL27870360

SCHEMBL27870360

CC(C=O)c1ccc(Nc2ccc(Br)cc2C(F)(F)F)cn1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.36
EGFR P00533 3/20 0.33
S1PR4 O95977 3/20 0.33
KDR P35968 1/20 0.33
HRH4 Q9H3N8 1/20 0.32
MPO P05164 1/20 0.32
ERBB2 P04626 1/20 0.32
ERBB3 P21860 1/20 0.32
ERBB4 Q15303 1/20 0.32
CNR2 P34972 1/20 0.32
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
DHODH Q02127 2/20 0.31
S1PR3 Q99500 2/20 0.31
TAS2R14 Q9NYV8 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
KDM1A O60341 2/20 0.30
SOS1 Q07889 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27853659 0.88 SCN1A (0.35) EGFRMPOERBB2ERBB3ERBB4
SCHEMBL27870327 0.86 RAB9A (0.38) CNR2DHODH
SCHEMBL185791 0.85 OPRM1 (0.38) OPRM1EGFRS1PR4KDRHRH4
SCHEMBL27870357 0.84 CNR2 (0.37) OPRM1EGFRS1PR4KDRMPO
SCHEMBL27870352 0.83 ALDH1A1 (0.42) EGFRDHODHTAS2R14
Trifluoroacetic Acid SCHEMBL185819 0.81 MPO (0.36) OPRM1EGFRS1PR4KDRHRH4
SCHEMBL184811 0.78 OPRM1 (0.44) OPRM1S1PR4MPOCNR2DHODH
SCHEMBL27853681 0.77 OPRM1 (0.39) OPRM1EGFRS1PR4KDRMPO
SCHEMBL185434 0.77 OPRM1 (0.35) OPRM1EGFRS1PR4KDRMPO
SCHEMBL184967 0.75 KIT (0.42) OPRM1EGFRKDRMPOCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102414177-A Compounds as bradykinin b1 antagonists BOEHRINGER INGELHEIM INT 2012-04-11 CN disclosed