SCHEMBL2787971

SCHEMBL2787971

C=CCN(CC=C)C1CC(NC(=O)O)(C(=O)NCc2ccc(Oc3ccc(OC)cc3C(F)(F)F)cc2)C1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
EPHX2 P34913 8/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
POLB P06746 1/20 0.36
PTPN7 P35236 2/20 0.35
DUSP3 P51452 2/20 0.35
P2RX7 Q99572 1/20 0.35
PPARG P37231 3/20 0.34
BTK Q06187 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13165656 0.88 BDKRB1 (0.40) CCR5NPSR1EPHX2POLBP2RX7
SCHEMBL2788429 0.88 NPSR1 (0.39) CCR5NPSR1EPHX2L3MBTL1POLB
SCHEMBL2808699 0.87 BTK (0.34) CCR5NPSR1EPHX2L3MBTL1POLB
SCHEMBL2787720 0.83 EPHX2 (0.41) EPHX2L3MBTL1POLBPTPN7DUSP3
SCHEMBL2786014 0.82 P2RX7 (0.41) EPHX2L3MBTL1POLBPTPN7DUSP3
SCHEMBL2790343 0.82 EPHX2 (0.41) EPHX2L3MBTL1POLBPTPN7DUSP3
SCHEMBL2787692 0.81 P2RX7 (0.42) EPHX2L3MBTL1POLBPTPN7DUSP3
SCHEMBL2788026 0.81 L3MBTL1 (0.42) EPHX2L3MBTL1POLBPTPN7DUSP3
SCHEMBL2785904 0.81 EPHX2 (0.40) EPHX2L3MBTL1POLBPTPN7DUSP3
SCHEMBL13165608 0.78 BDKRB1 (0.37) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097374-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed