SCHEMBL27883

SCHEMBL27883

COc1ccc([CH]c2ccc(OC)cc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.65
CA1 P00915 1/20 0.65
CA2 P00918 1/20 0.65
CA7 P43166 1/20 0.65
CA9 Q16790 1/20 0.65
CA14 Q9ULX7 1/20 0.65
ALDH1A1 P00352 3/20 0.64
CYP2A6 P11509 1/20 0.64
KDM4E B2RXH2 4/20 0.61
CYP3A4 P08684 2/20 0.61
LMNA P02545 2/20 0.61
TP53 P04637 1/20 0.61
TSHR P16473 1/20 0.61
TRPA1 O75762 1/20 0.58
RELA Q04206 1/20 0.58
CYP1A2 P05177 3/20 0.56
CYP1A1 P04798 3/20 0.56
CYP1B1 Q16678 3/20 0.56
ESR1 P03372 2/20 0.56
PTGS2 P35354 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18240595 0.90 RELA (0.75) CA12CA1CA2CA7CA9
SCHEMBL290332 0.90 TRPA1 (0.75) CA12CA1CA2CA7CA9
SCHEMBL14880493 0.88 AHR (0.57) CA12CA1CA2CA7CA9
SCHEMBL14880245 0.88 NFE2L2 (0.76) CA12CA1CA2CA7CA9
SCHEMBL11090821 0.86 CYP1A2 (0.77) CA12CA1CA2CA7CA9
SCHEMBL698571 0.82 CYP1A1 (0.58) CA12CA1CA2CA7CA9
SCHEMBL29016917 0.82 AHR (0.72) CA12CA1CA2CA7CA9
SCHEMBL13790336 0.82 RELA (0.81) ALDH1A1KDM4ECYP3A4LMNATP53
SCHEMBL4881152 0.82 RELA (0.81) ALDH1A1KDM4ECYP3A4LMNATP53
SCHEMBL631998 0.82 RELA (0.81) ALDH1A1KDM4ECYP3A4LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6487 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240158417-A1 SUBSTITUTED HETEROCYCLIC FUSED CYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF GENFLEET THERAPEUTICS (SHANGHAI) INC. (CN) 2024-05-16 US claimed
EP-4328229-A2 SUBSTITUTED HETEROCYCLIC FUSED CYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF Genfleet Therapeutics (Shanghai) Inc. (CN) 2024-02-28 EP claimed
CN-112010889-B Preparation method of 4-hydroxy-2-azetidinone compound 中国科学院上海营养与健康研究所 2023-09-19 CN claimed
WO-2023151188-A1 GREEN SYNTHESIS METHOD OF ANTIVIRAL DRUG INTERMEDIATE 上海皓元医药股份有限公司 2023-08-17 WO claimed
CN-114671798-B Green synthesis method of antiviral drug intermediate 上海皓元医药股份有限公司 2022-08-16 CN claimed
CN-114671798-A Green synthesis method of antiviral drug intermediate 上海皓元医药股份有限公司 2022-06-28 CN claimed
EP-3053944-B1 METHOD FOR PRODUCING POLYALKYLENE GLYCOL DERIVATIVE HAVING AMINO GROUP AT END, POLYMERIZATION INITIATOR FOR USE IN THE SAME, AND ALCOHOL COMPOUND AS RAW MATERIAL FOR THE POLYMERIZATION INITIATOR SHINETSU CHEMICAL CO (JP) 2021-10-06 EP claimed
CN-112010889-A Preparation method of 4-hydroxy-2-azetidinone compound 中国科学院上海营养与健康研究所 2020-12-01 CN claimed
US-20200223860-A1 THE TOTAL SYNTHESIS OF GLUCOSEPANE AND RELATED CHEMICAL REACTIONS, COMPOUNDS AND COMPOSITIONS AND OBTAINED THEREFROM AND METHODS OF TREATMENT UNIV YALE (US) 2020-07-16 US claimed
CN-110669058-A Tricyclic quinolone carboxylic acid and preparation method thereof 江西农业大学 2020-01-10 CN claimed
US-4145538-A 3-Carbamyloxymethyl-cephalosporins ELI LILLY AND COMPANY (US) 1979-03-20 US claimed
US-4118483-A Peptides having gonadoliberin activity and process for their manufacture HOECHST AKTIENGESELLSCHAFT (DE) 1978-10-03 US claimed
US-4117117-A TRIDECAPETIDE HAVING GASTRIN EFFECT MAX PLANCK-GESELLSCHAFT ZUR FORDERUNG DER WISSENSCHAFTEN (DE) 1978-09-26 US claimed
US-4092306-A Oxidation of hydrazones to the corresponding diazo compounds in the presence of a phase transfer and an oxidation catalyst which is iodine, an iodide or an iodonium salt GLAXO LABORATORIES LIMITED (EN) 1978-05-30 US claimed
US-4092474-A Cephalosporins having a metaloxy group in 3-substituent SHIONOGI & CO., LTD. (JA) 1978-05-30 US claimed
US-4009159-A PENICILLINS FUJISAWA PHARMACEUTICAL CO., LTD. (JA) 1977-02-22 US claimed
US-3953437-A Process of preparing cephalosporanic acid ester derivatives YAMANOUCHI PHARMACEUTICAL CO., LTD. (JA) 1976-04-27 US claimed
US-3944545-A Process for preparing desacetoxycephalosporins ELI LILLY AND COMPANY (US) 1976-03-16 US claimed
US-3935198-A BY HEATING THE PENICILLIN SULFOXIDE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JA) 1976-01-27 US claimed
US-3932465-A ANTIBIOTIC CIBA-GEIGY CORPORATION (US) 1976-01-13 US claimed