SCHEMBL278963

SCHEMBL278963

C=C(/N=C/c1cc(F)ccc1OC1CCSCC1)O[Si](C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 2/20 0.34
ITGB2 P05107 1/20 0.32
ICAM1 P05362 1/20 0.32
ITGAL P20701 1/20 0.32
RBP4 P02753 1/20 0.31
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL275957 1.00 FPR2 (0.34) FPR2ITGB2ICAM1ITGALRBP4
SCHEMBL274398 0.90 PDE4D (0.36)
SCHEMBL279473 0.90 PDE4D (0.36)
SCHEMBL274953 0.89 PTGDR2 (0.36)
SCHEMBL279471 0.89 PTGDR2 (0.36)
SCHEMBL279161 0.88 SYK (0.39)
SCHEMBL276376 0.88 SYK (0.39)
SCHEMBL274636 0.87 HPGD (0.38) FPR2IDO1
SCHEMBL279174 0.87 HPGD (0.38) FPR2IDO1
SCHEMBL8043283 0.80 ERN1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8134001-B2 Spiroindolinone derivatives HOFFMANN-LA ROCHE INC. (US) 2012-03-13 US disclosed
US-20090156610-A1 Spiroindolinone Derivatives DING QINGJIE 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156610-A1 Spiroindolinone Derivatives SDHA, AR, XPOT FPR2 4631/4885ITGB2 1997/4885ICAM1 4727/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.