SCHEMBL27899243

SCHEMBL27899243

CC(C)(CNc1ncc(COC=O)cn1)c1ccc(F)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 6/20 0.38
HDAC3 O15379 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
ME2 P23368 1/20 0.34
ME1 P48163 1/20 0.34
ME3 Q16798 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CACNA1G O43497 1/20 0.32
PTK2 Q05397 1/20 0.31
MAPK14 Q16539 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2562645 0.76 HDAC6 (0.41) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL2560721 0.75 VNN1 (0.47) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL2566143 0.74 VNN1 (0.49) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL19942194 0.73 VNN1 (0.39) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL2560278 0.72 HDAC3 (0.53) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL17080669 0.70 HDAC6 (0.39) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL12288597 0.69 VNN1 (0.44) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL22975115 0.68 KMT2A (0.46) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL2560412 0.68 GPR55 (0.45) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL18466466 0.68 HDAC3 (0.48) VNN1HDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105712974-A Certain Amino-Pyridazines, Compositions Thereof, And Methods Of Their Use 赛特凯恩蒂克公司 2016-06-29 CN disclosed
CN-103025331-B Certain amino-pyrimidines, compositions thereof and methods of use thereof CYTOKINETICS, INC. (US) 2016-03-02 CN disclosed
CN-103025331-A Certain amino-pyrimidines, compositions thereof and methods of use thereof CYTOKINETICS INC 2013-04-03 CN disclosed