SCHEMBL2790195

SCHEMBL2790195

COCCCn1c(C2CCCN(C(=O)C[C@H](N)Cc3ccc(-c4ccc5c(c4)CC(=O)N5)cc3)C2)cc2c(F)cccc21

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.35
SMYD3 Q9H7B4 8/20 0.35
CNR2 P34972 1/20 0.34
CFD P00746 2/20 0.34
CDK2 P24941 2/20 0.33
CRBN Q96SW2 1/20 0.33
PADI4 Q9UM07 1/20 0.33
CTSC P53634 1/20 0.32
ABCB1 P08183 1/20 0.32
DPP4 P27487 1/20 0.32
LIPG Q9Y5X9 1/20 0.32
CDK1 P06493 1/20 0.32
KIT P10721 1/20 0.32
KDR P35968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2791483 0.91 CNR2 (0.33) CNR2CFDCTSCDPP4
SCHEMBL741417 0.89 CFD (0.36) AKT1SMYD3CFDCDK2CRBN
SCHEMBL741416 0.89 CFD (0.36) AKT1SMYD3CFDCDK2CRBN
SCHEMBL2789341 0.87 CNR2 (0.37) CNR2CFDDPP4
SCHEMBL2789943 0.86 AKT1 (0.36) AKT1SMYD3CNR2CDK2CTSC
SCHEMBL2791998 0.86 CNR2 (0.35) CNR2CFDDPP4
SCHEMBL2792440 0.85 CNR2 (0.36) CNR2CFDDPP4
SCHEMBL741966 0.84 AKT1 (0.36) AKT1SMYD3CFDCDK2CRBN
SCHEMBL742052 0.84 AKT1 (0.36) AKT1SMYD3CFDCDK2CRBN
SCHEMBL742026 0.84 CFD (0.37) SMYD3CFDCRBNPADI4CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO claimed
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed