SCHEMBL742052

SCHEMBL742052

COCCCn1c(C2CCCN(C(=O)CC(N)Cc3ccc(-c4ccc5c(c4)CC(=O)N5)cc3)C2)nc2c(C)cccc21

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 2/20 0.36
GRIA1 P42261 1/20 0.35
CACNG8 Q8WXS5 1/20 0.35
PADI4 Q9UM07 3/20 0.35
SMYD3 Q9H7B4 8/20 0.34
BTK Q06187 1/20 0.33
CDK2 P24941 1/20 0.33
CPT2 P23786 2/20 0.33
CPT1A P50416 2/20 0.33
CRBN Q96SW2 1/20 0.33
CFD P00746 1/20 0.32
NPY1R P25929 1/20 0.32
CPT1B Q92523 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741966 1.00 AKT1 (0.36) AKT1GRIA1CACNG8PADI4SMYD3
SCHEMBL741416 0.93 CFD (0.36) AKT1PADI4SMYD3CDK2CPT2
SCHEMBL741417 0.93 CFD (0.36) AKT1PADI4SMYD3CDK2CPT2
SCHEMBL741160 0.91 BTK (0.31) BTKCFDNPY1R
SCHEMBL741161 0.91 BTK (0.31) BTKCFDNPY1R
SCHEMBL742030 0.90 NSD2 (0.36) PADI4
SCHEMBL742029 0.90 NSD2 (0.36) PADI4
SCHEMBL741987 0.89 SMYD3 (0.35) PADI4SMYD3BTKCFDNPY1R
SCHEMBL741986 0.89 SMYD3 (0.35) PADI4SMYD3BTKCFDNPY1R
SCHEMBL740294 0.88 CFD (0.37) PADI4SMYD3CPT2CPT1ACRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed