SCHEMBL2790486

SCHEMBL2790486

Cc1oc(C(N)=O)c2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.41
ALDH1A1 P00352 3/20 0.41
POLB P06746 2/20 0.40
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
TEAD1 P28347 1/20 0.40
YAP1 P46937 1/20 0.40
TEAD4 Q15561 1/20 0.40
TEAD2 Q15562 1/20 0.40
MAPT P10636 3/20 0.38
AHR P35869 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
GAA P10253 1/20 0.38
HSD17B10 Q99714 3/20 0.37
TP53 P04637 2/20 0.37
MAPK10 P53779 2/20 0.37
TSHR P16473 2/20 0.37
CYP2C19 P33261 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7861729 0.82 MCL1 (0.49) KDM4EALDH1A1KMT2AMAPTNPC1
SCHEMBL114253 0.82 GAA (0.47) KDM4EALDH1A1POLBKMT2AMAPT
SCHEMBL9433289 0.78 ALDH1A1 (0.41) KDM4EALDH1A1POLBKMT2ATEAD1
SCHEMBL9399721 0.77 SMN1; SMN2 (0.38) KDM4EALDH1A1KMT2AMEN1MAPT
SCHEMBL27917704 0.77 KDM4E (0.40) KDM4EALDH1A1KMT2AMEN1MAPT
SCHEMBL353910 0.73 KCNH2 (0.58) KDM4EALDH1A1KMT2AMEN1TEAD1
SCHEMBL2607276 0.72 CYP1A2 (0.47) KDM4EALDH1A1MAPTAHRSMN1; SMN2
SCHEMBL9433908 0.72 IRAK4 (0.46) KDM4EALDH1A1KMT2AMEN1TEAD1
SCHEMBL27494718 0.71 PTPN1 (0.46) KMT2AMEN1TEAD1YAP1TEAD4
SCHEMBL7574372 0.69 CAPN1 (0.54) KDM4EALDH1A1KMT2AMEN1TEAD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2161266-A1 Benzofuran derivatives as orexin receptor antagonists EVOTEC Neurosciences GmbH (DE) 2010-03-10 EP disclosed