SCHEMBL27907697

SCHEMBL27907697

COc1ccc(Nc2ncnc3ccc(-c4cccc(C#N)c4)cc23)cc1Cl

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.62
ABCG2 Q9UNQ0 2/20 0.62
CYP1A2 P05177 5/20 0.61
HSD17B10 Q99714 5/20 0.61
CYP3A4 P08684 4/20 0.61
CLK4 Q9HAZ1 4/20 0.61
ALDH1A1 P00352 4/20 0.61
LMNA P02545 4/20 0.61
TSHR P16473 4/20 0.61
MAPK1 P28482 4/20 0.61
USP2 O75604 3/20 0.61
CYP2C19 P33261 2/20 0.61
CYP2D6 P10635 2/20 0.61
HIF1A Q16665 2/20 0.61
CYP2C9 P11712 4/20 0.58
BRAF P15056 11/20 0.57
RAF1 P04049 10/20 0.57
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
TP53 P04637 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28801394 0.86 BRAF (0.67) EGFRCYP1A2HSD17B10CYP3A4CLK4
SCHEMBL27890908 0.85 RAF1 (0.70) EGFRABCG2BRAFRAF1ERBB2
SCHEMBL28801011 0.82 RAF1 (0.60) EGFRBRAFRAF1ERBB2
SCHEMBL27890907 0.82 BRAF (0.59) EGFRCYP1A2HSD17B10CYP3A4CLK4
SCHEMBL27907718 0.81 RAF1 (0.60) EGFRALDH1A1BRAFRAF1ERBB2
SCHEMBL27907693 0.81 BRAF (0.71) EGFRBRAFRAF1ERBB2
SCHEMBL27987180 0.81 RAF1 (0.72) EGFRABCG2BRAFRAF1ERBB2
SCHEMBL27986782 0.79 EGFR (0.61) EGFRBRAFRAF1ERBB2ERBB4
SCHEMBL27907705 0.79 MAP4K1 (0.49) ABCG2ALDH1A1LMNABRAFMEN1
SCHEMBL17845962 0.78 RAF1 (0.59) EGFRABCG2BRAFRAF1ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102924387-A 4-(3-chloro-4-methoxyanilino)-6-(3,4-substituted phenyl)quinazoline and salts thereof, preparation method and applications HUANG WEIYAN 2013-02-13 CN claimed
CN-102924387-B 4-(3-chloro-4-methoxyanilino)-6-(3,4-substituted phenyl)quinazoline and salts thereof, preparation method and applications HUANG WEIYAN 2015-07-01 CN disclosed
CN-102924387-A 4-(3-chloro-4-methoxyanilino)-6-(3,4-substituted phenyl)quinazoline and salts thereof, preparation method and applications HUANG WEIYAN 2013-02-13 CN disclosed