SCHEMBL27908400

SCHEMBL27908400

O=C(F)c1cc(-c2ccccc2)ccc1[N+](=O)[O-]

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.51
CRHR2 Q13324 1/20 0.51
ABCB1 P08183 7/20 0.49
ABCC1 P33527 6/20 0.49
KCNMA1 Q12791 1/20 0.49
POLB P06746 1/20 0.45
MAPK1 P28482 1/20 0.45
ACMSD Q8TDX5 2/20 0.45
DHFR P00374 1/20 0.45
HNF4A P41235 1/20 0.45
MCL1 Q07820 1/20 0.45
DTYMK P23919 1/20 0.44
ALDH1A1 P00352 2/20 0.44
TDP1 Q9NUW8 1/20 0.43
ALOX5 P09917 1/20 0.43
IKBKB O14920 1/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27985266 0.87 DTYMK (0.58) CRHBPCRHR2ABCB1ABCC1KCNMA1
SCHEMBL25302339 0.84 ABCB1 (0.52) CRHBPCRHR2ABCB1ABCC1KCNMA1
SCHEMBL8372988 0.84 CRHBP (0.51) CRHBPCRHR2ABCB1ABCC1KCNMA1
SCHEMBL8372989 0.82 CRHBP (0.53) CRHBPCRHR2ABCB1ABCC1KCNMA1
Acetamide SCHEMBL2368476 0.80 DTYMK (0.51) CRHBPCRHR2ABCB1ABCC1KCNMA1
SCHEMBL31232900 0.79 CRHBP (0.46) CRHBPCRHR2ABCB1ABCC1KCNMA1
SCHEMBL3325012 0.77 ALDH1A1 (0.63) ALDH1A1TDP1MAPT
SCHEMBL1663325 0.77 CRHBP (0.63) CRHBPCRHR2ABCB1ABCC1KCNMA1
SCHEMBL8365480 0.77 ABCB1 (0.49) CRHBPCRHR2ABCB1ABCC1KCNMA1
SCHEMBL15847247 0.77 ALDH1A1 (0.51) ABCB1ABCC1POLBALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101970429-B 2-amino-quinoline derivatives useful as inhibitors of beta-secretase (bace) JANSSEN PHARMACEUTICA NV 2013-05-29 CN disclosed