SCHEMBL27913624

SCHEMBL27913624

CC(C)(C)NCc1ccc(OC(F)(F)F)c(Cl)c1.NC(=O)c1ccncc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN3A Q9NY46 7/20 0.48
SCN1A P35498 2/20 0.45
SCN5A Q14524 2/20 0.45
SCN9A Q15858 2/20 0.45
SCN2A Q99250 2/20 0.45
SCN8A Q9UQD0 2/20 0.45
SCN10A Q9Y5Y9 2/20 0.45
KCNH2 Q12809 1/20 0.45
CSF1R P07333 1/20 0.44
ALPL P05186 1/20 0.41
AKT1 P31749 1/20 0.41
ROCK2 O75116 1/20 0.41
KMO O15229 1/20 0.39
LMNA P02545 2/20 0.39
MRGPRX4 Q96LA9 1/20 0.39
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28093912 0.89 SCN3A (0.46) SCN3ASCN1ASCN5ASCN9ASCN2A
SCHEMBL27913628 0.88 P2RX7 (0.45) SCN3ASCN1ASCN5ASCN9ASCN2A
SCHEMBL27913866 0.86 CTSD (0.40) SCN3ASCN5ASCN9AALPLROCK2
Pyrazinamide SCHEMBL28833282 0.85 SCN3A (0.44) SCN3ASCN1ASCN5ASCN9ASCN2A
SCHEMBL27913648 0.82 AURKA (0.53) ROCK2AURKARPS6KB1AURKB
SCHEMBL28093971 0.78 P2RX7 (0.43) SCN3ASCN1ASCN5ASCN9ASCN2A
SCHEMBL27931776 0.76 VNN1 (0.46) AKT1AURKARPS6KB1AURKB
SCHEMBL27913577 0.76 VNN1 (0.53) AURKARPS6KB1AURKB
SCHEMBL27931758 0.76 HDAC3 (0.40) SCN9AROCK2
SCHEMBL28833323 0.76 CTSD (0.39) SCN3ASCN1ASCN5ASCN9ASCN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103249721-A Arylamine Derivatives as TTX-S Blockers RAQUALIA PHARMA INC 2013-08-14 CN claimed
CN-103249721-A Arylamine Derivatives as TTX-S Blockers RAQUALIA PHARMA INC 2013-08-14 CN disclosed