SCHEMBL27923217

SCHEMBL27923217

COc1ccc(CN2CCCCCC2=O)c(OC)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.56
KDM4E B2RXH2 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
ALDH1A1 P00352 2/20 0.47
TSHR P16473 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47
MTNR1A P48039 1/20 0.47
MTNR1B P49286 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8373325 0.95 MTNR1A (0.52) ACHEKDM4EMEN1KMT2AALDH1A1
SCHEMBL10640944 0.89 KDM4E (0.53) KDM4EMEN1KMT2AALDH1A1TSHR
SCHEMBL2227533 0.82 HDAC3 (0.50) KDM4EMEN1KMT2AALDH1A1TSHR
SCHEMBL27396041 0.81 APLNR (0.51) KDM4EMEN1KMT2AALDH1A1TSHR
SCHEMBL20303832 0.80 L3MBTL1 (0.67) MEN1KMT2AALDH1A1HDAC1HDAC6
SCHEMBL17185001 0.80 ACHE (0.49) ACHEKDM4EALDH1A1HDAC1HDAC6
SCHEMBL22993631 0.80 ACHE (0.48) ACHEKMT2AALDH1A1HDAC6MTNR1A
SCHEMBL17184827 0.80 KDM4E (0.50) ACHEKDM4EKMT2AHDAC6ADRA1D
SCHEMBL8373324 0.79 MTNR1A (0.50) KDM4EMEN1KMT2AALDH1A1MTNR1A
SCHEMBL3459387 0.79 L3MBTL1 (0.64) MEN1KMT2AALDH1A1HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101090902-B Cgrp receptor antagonists MERCK SHARP & DOHME 2013-05-29 CN disclosed